SCHEMBL4046398

SCHEMBL4046398

CC(Cc1ccc(Br)cc1)NC(=O)C(F)(F)F

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACACB O00763 10/20 0.57
ESR1 P03372 1/20 0.50
KCNH2 Q12809 1/20 0.50
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
KMT2A Q03164 2/20 0.46
SIGMAR1 Q99720 1/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8986825 0.86 ESR1 (0.54) ACACBESR1KCNH2NPC1RAB9A
SCHEMBL8986819 0.86 ESR1 (0.54) ACACBESR1KCNH2NPC1RAB9A
SCHEMBL11959175 0.86 ACACB (0.56) ACACBESR1KCNH2NPC1RAB9A
SCHEMBL4474242 0.84 CYP1A2 (0.51) ACACBESR1KCNH2NPC1RAB9A
SCHEMBL6540778 0.84 CYP1A2 (0.51) ACACBESR1KCNH2NPC1RAB9A
SCHEMBL6677150 0.84 CYP1A2 (0.51) ACACBESR1KCNH2NPC1RAB9A
SCHEMBL6801338 0.84 ESR1 (0.50) ACACBESR1KCNH2NPC1RAB9A
SCHEMBL11695904 0.84 ESR1 (0.57) ACACBESR1KCNH2NPC1RAB9A
SCHEMBL11695897 0.84 ESR1 (0.57) ACACBESR1KCNH2NPC1RAB9A
SCHEMBL12204087 0.84 ACACB (0.57) ACACBESR1KCNH2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011124093-A1 BICYCLIC QUINOLONE COMPOUNDS, PREPARATION METHODS AND USES THEREOF 山东轩竹医药科技有限公司 (CN) 2011-10-13 WO disclosed
WO-2009103478-A1 PYRIDONE AND PYRIDAZINONE DERIVATIVES AS MCH ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-08-27 WO disclosed