SCHEMBL4046832

SCHEMBL4046832

N#Cc1cccc2c1COCO2

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.37
ABCG2 Q9UNQ0 1/20 0.37
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
CYP11B1 P15538 5/20 0.34
CYP11B2 P19099 5/20 0.34
HTR2A P28223 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.33
SIRT1 Q96EB6 1/20 0.33
TSHR P16473 1/20 0.32
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30969397 0.77 ABCG2 (0.33) ABCG2HTR2AALDH1A1SIRT2SIRT1
SCHEMBL17069064 0.77 ABCG2 (0.44) TRPA1ABCG2NPC1RAB9ACYP11B1
SCHEMBL29361235 0.73 ABCG2 (0.39) ABCG2ALDH1A1TSHR
SCHEMBL7481318 0.73 ABCG2 (0.39) ABCG2ALDH1A1TSHR
SCHEMBL6955296 0.73 ABCG2 (0.39) ABCG2ALDH1A1TSHR
SCHEMBL31634143 0.73 ABCG2 (0.39) ABCG2HTR2ATSHR
SCHEMBL12043582 0.73 MAP3K14 (0.41) ABCG2KDM4EALDH1A1TSHR
SCHEMBL14304553 0.73 ITGB2 (0.39) TRPA1NPC1RAB9ATSHR
SCHEMBL6928146 0.73 ABCG2 (0.39) ABCG2TSHR
SCHEMBL23668349 0.70 ABCG2 (0.37) ABCG2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010532-A1 TRYCLIC NITROGEN CONTAINING COMPOUNDS AND THEIR USE AS ANTIBACTERIALS Glaxo Group Limited (GB) 2009-01-07 EP claimed
WO-2007122258-A1 TRYCLIC NITROGEN CONTAINING COMPOUNDS AND THEIR USE AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2007-11-01 WO claimed
CN-116180112-A Method for electrochemical synthesis of aryl nitrile by using dialkyl aryl phosphate 河南大学 2023-05-30 CN disclosed