SCHEMBL4046909

SCHEMBL4046909

COc1cc(Nc2nc(N)n(-c3ccccc3F)n2)cc(OC)c1

nearest known ligand 0.72

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 9/20 0.72
BACE1 P56817 3/20 0.55
AXL P30530 1/20 0.48
KIT P10721 2/20 0.46
IRAK4 Q9NWZ3 2/20 0.46
AURKA O14965 1/20 0.46
JAK2 O60674 1/20 0.46
SLC29A2 Q14542 1/20 0.43
SLC29A1 Q99808 1/20 0.43
JAK1 P23458 2/20 0.40
TYK2 P29597 2/20 0.40
JAK3 P52333 1/20 0.40
CYP1A1 P04798 1/20 0.40
CYP1B1 Q16678 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPK1 P28482 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12780526 0.87 FLT3 (0.62) FLT3BACE1AXLKITIRAK4
SCHEMBL4039143 0.86 FLT3 (0.80) FLT3BACE1AXLKITIRAK4
SCHEMBL4044001 0.84 FLT3 (1.00) FLT3BACE1AXLKITIRAK4
SCHEMBL2088273 0.82 FLT3 (0.67) FLT3BACE1AXLKITIRAK4
SCHEMBL4040306 0.79 AXL (0.76) FLT3AXLKITIRAK4AURKA
SCHEMBL28335490 0.78 FLT3 (0.61) FLT3BACE1AXLKITAURKA
SCHEMBL4036286 0.76 FLT3 (0.64) FLT3AXLKITIRAK4AURKA
SCHEMBL2088150 0.76 FLT3 (0.63) FLT3BACE1AXLKITIRAK4
SCHEMBL3963633 0.75 FLT3 (0.61) FLT3BACE1AXLKITAURKA
SCHEMBL4043057 0.75 BACE1 (0.58) FLT3BACE1AXLKITIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562589-B1 DIAMINOTRIAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2009-01-07 EP disclosed