SCHEMBL4047067

SCHEMBL4047067

COc1ccc2nccc(N3CCC(N(C(=O)O)C(CNC(=O)C(F)(F)F)C(C)(C)C)C3)c2n1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP8B1 Q9UNU6 2/20 0.49
HRH4 Q9H3N8 3/20 0.39
HRH3 Q9Y5N1 3/20 0.39
CYP2C19 P33261 1/20 0.38
PIK3CA P42336 1/20 0.38
SLC2A1 P11166 1/20 0.37
KCNH2 Q12809 7/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3168285 0.84 CYP8B1 (0.49) CYP8B1HRH4HRH3CYP2C19PIK3CA
SCHEMBL13527137 0.80 CYP8B1 (0.47) CYP8B1HRH4HRH3CYP2C19PIK3CA
SCHEMBL3167861 0.78 CYP8B1 (0.49) CYP8B1SLC2A1KCNH2
SCHEMBL5905803 0.75 CYP8B1 (0.50) CYP8B1CYP2C19PIK3CASLC2A1KCNH2
SCHEMBL3162808 0.75 CYP8B1 (0.49) CYP8B1CYP2C19PIK3CASLC2A1KCNH2
SCHEMBL3177584 0.74 MAP4K4 (0.52) CYP8B1CYP2C19PIK3CAKCNH2
SCHEMBL3162840 0.73 CYP8B1 (0.47) CYP8B1HRH4HRH3CYP2C19PIK3CA
SCHEMBL4071024 0.73 CYP8B1 (0.45) CYP8B1CYP2C19KCNH2
SCHEMBL1224565 0.72 CYP8B1 (0.53) CYP8B1CYP2C19PIK3CAKCNH2
SCHEMBL10078646 0.72 CYP8B1 (0.53) CYP8B1CYP2C19PIK3CAKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773343-A4 ANTIBACTERIAL AGENTS GLAXO GROUP LTD (GB) 2009-05-13 EP disclosed
EP-1773343-A1 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2007-04-18 EP disclosed
WO-2006017326-A1 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2006-02-16 WO disclosed