SCHEMBL4048825

SCHEMBL4048825

O=C1CNC(=O)N1[C@H]1C[C@@H](n2cnc3c(N(CO)CCc4ccccc4)nc(Cl)nc32)[C@H](O)[C@@H]1O

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.39
ADORA3 P0DMS8 4/20 0.39
ADORA2A P29274 4/20 0.38
NT5E P21589 5/20 0.37
TMIGD3 P0DMS9 3/20 0.36
HTR2C P28335 3/20 0.36
HTR2B P41595 3/20 0.36
HTR3A P46098 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1412120 0.81 ADORA2A (0.33) ADORA1ADORA3ADORA2A
SCHEMBL1412466 0.77 ADORA1 (0.61) ADORA1ADORA3ADORA2A
SCHEMBL3891540 0.77 NT5E (0.38) ADORA1ADORA3ADORA2ANT5ETMIGD3
SCHEMBL1412222 0.75 ADORA2A (0.55) ADORA1ADORA3ADORA2ANT5E
Acetic Acid SCHEMBL6838891 0.69 NT5E (0.43) ADORA1ADORA3ADORA2ANT5E
SCHEMBL6838896 0.67 NT5E (0.41) ADORA1ADORA3ADORA2ANT5E
SCHEMBL4374282 0.66 ADORA2A (0.42) ADORA3ADORA2A
SCHEMBL1412158 0.66 ADORA2A (0.54) ADORA1ADORA3ADORA2A
SCHEMBL1412256 0.64 ADORA2A (0.48) ADORA1ADORA3ADORA2A
SCHEMBL17150935 0.64 NT5E (0.41) ADORA1ADORA3ADORA2ANT5ETMIGD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2018388-A2 BISADENOSINE COMPOUNDS AS ADENOSINE A2A RECEPTOR AGONISTS Novartis AG (CH) 2009-01-28 EP disclosed
WO-2007121924-A2 BISADENOSINE COMPOUNDS AS ADENOSINE A2A RECEPTOR AGONISTS NOVARTIS AG (CH) 2007-11-01 WO disclosed