SCHEMBL4056601

SCHEMBL4056601

CN1CCN(c2cc(-c3cccc(C#N)c3)ncn2)CC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 3/20 0.67
CYP1A2 P05177 9/20 0.58
ALDH1A1 P00352 4/20 0.58
CYP3A4 P08684 3/20 0.58
USP2 O75604 2/20 0.58
CLK4 Q9HAZ1 2/20 0.58
MEN1 O00255 1/20 0.58
KMT2A Q03164 1/20 0.58
HIF1A Q16665 1/20 0.58
LRRK2 Q5S007 2/20 0.58
GRM5 P41594 2/20 0.58
DPP4 P27487 2/20 0.57
HSD17B10 Q99714 4/20 0.57
ALOX15 P16050 3/20 0.57
CYP2C19 P33261 3/20 0.57
KDM4E B2RXH2 1/20 0.55
GLA P06280 1/20 0.55
MAPT P10636 1/20 0.55
HPGD P15428 1/20 0.55
TSHR P16473 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL604430 0.81 HRH4 (0.76) HRH4HTR1AADRA2AADRA2CHTR1D
Hydrochloric Acid SCHEMBL11785742 0.80 HRH4 (0.97) HRH4CYP1A2ALDH1A1DPP4HSD17B10
SCHEMBL4061028 0.78 HRH4 (0.67) HRH4CYP1A2ALDH1A1DPP4HSD17B10
SCHEMBL2384302 0.77 HRH4 (0.69) HRH4CYP1A2ALDH1A1CYP3A4USP2
SCHEMBL28302301 0.75 LRRK2 (0.62) CYP1A2CYP3A4LRRK2GRM5DPP4
SCHEMBL10268958 0.74 HRH4 (0.55) HRH4CYP1A2ALDH1A1CYP3A4USP2
SCHEMBL12331397 0.74 GRM5 (0.62) CYP1A2ALDH1A1CYP3A4USP2CLK4
SCHEMBL9792862 0.72 GRM5 (0.64) CYP1A2ALDH1A1CYP3A4USP2CLK4
Hydrochloric Acid SCHEMBL11786310 0.72 HRH4 (0.72) HRH4CYP1A2ALDH1A1MEN1KMT2A
SCHEMBL9792981 0.71 GRM5 (0.62) CYP1A2ALDH1A1CYP3A4USP2CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009035671-A1 SUBSTITUTED NITROGEN-CONTAINING HETEROARYL DERIVATIVES USEFUL AS MODULATORS OF THE HISTAMINE H4 RECEPTOR JANSSEN PHARMACEUTICA N.V. (BE) 2009-03-19 WO claimed