SCHEMBL4058428

SCHEMBL4058428

CC(C)C(CO)Nc1nc(Nc2ccc(S(C)(=O)=O)cc2)ncc1Br

nearest known ligand 0.67

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 19/20 0.67
CDK2 P24941 19/20 0.67
KDR P35968 16/20 0.67
CA2 P00918 2/20 0.67
CDK4 P11802 2/20 0.67
CDK7 P50613 2/20 0.67
CDK9 P50750 2/20 0.67
CCNT1 O60563 1/20 0.67
CCND1 P24385 1/20 0.67
CCNH P51946 1/20 0.67
CCNB1 P14635 2/20 0.66
CCNE1 P24864 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4058417 1.00 CDK1 (0.67) CDK1CDK2KDRCA2CDK4
SCHEMBL4057630 0.92 CDK1 (0.80) CDK1CDK2KDRCA2CDK4
SCHEMBL4063258 0.92 CDK1 (0.80) CDK1CDK2KDRCA2CDK4
SCHEMBL13648671 0.92 CDK1 (0.67) CDK1CDK2KDRCA2CDK4
SCHEMBL4064917 0.91 CDK1 (0.66) CDK1CDK2KDRCA2CDK4
SCHEMBL13648674 0.91 CDK1 (0.66) CDK1CDK2KDRCA2CDK4
SCHEMBL4063631 0.90 CDK1 (0.65) CDK1CDK2KDRCA2CDK4
SCHEMBL4062664 0.90 CDK1 (0.65) CDK1CDK2KDRCA2CDK4
SCHEMBL4064827 0.90 CDK1 (0.65) CDK1CDK2KDRCA2CDK4
SCHEMBL4058222 0.88 CDK1 (0.63) CDK1CDK2KDRCA2CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392662-B1 CDK INHIBITING PYRIMIDINES, PRODUCTION THEREOF AND THEIR USE AS MEDICAMENTS BAYER SCHERING PHARMA AG (DE) 2009-01-07 EP claimed
EP-1392662-B1 CDK INHIBITING PYRIMIDINES, PRODUCTION THEREOF AND THEIR USE AS MEDICAMENTS BAYER SCHERING PHARMA AG (DE) 2009-01-07 EP disclosed