SCHEMBL4060010

SCHEMBL4060010

Cc1cc2c(-c3ccc(S(=O)(=O)NC4CC[S+]([O-])CC4)cc3)ccnc2[nH]1

nearest known ligand 0.75

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 19/20 0.75
CHUK O15111 19/20 0.75
ROCK1 Q13464 1/20 0.58
AURKB Q96GD4 1/20 0.52
AURKAIP1 Q9NWT8 1/20 0.52
KIT P10721 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4052716 0.92 IKBKB (0.65) IKBKBCHUKROCK1AURKBAURKAIP1
SCHEMBL3418269 0.89 IKBKB (0.81) IKBKBCHUKROCK1AURKBAURKAIP1
SCHEMBL3417539 0.89 IKBKB (0.79) IKBKBCHUKROCK1AURKBAURKAIP1
SCHEMBL3418133 0.88 IKBKB (0.78) IKBKBCHUKROCK1AURKBAURKAIP1
SCHEMBL14154259 0.87 IKBKB (0.76) IKBKBCHUKROCK1AURKBAURKAIP1
SCHEMBL3417920 0.87 IKBKB (0.76) IKBKBCHUKROCK1AURKBAURKAIP1
SCHEMBL3412681 0.86 IKBKB (1.00) IKBKBCHUKROCK1AURKBAURKAIP1
SCHEMBL3417228 0.86 IKBKB (0.78) IKBKBCHUKROCK1KIT
SCHEMBL4052036 0.85 IKBKB (0.62) IKBKBCHUK
SCHEMBL3412679 0.85 IKBKB (0.83) IKBKBCHUKROCK1AURKBAURKAIP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009112475-A1 PYRROLO [2, 3-B] PYRIDIN DERIVATIVES AS IKK2 INHIBITORS GLAXO GROUP LIMITED (GB) 2009-09-17 WO claimed
WO-2009112475-A1 PYRROLO [2, 3-B] PYRIDIN DERIVATIVES AS IKK2 INHIBITORS GLAXO GROUP LIMITED (GB) 2009-09-17 WO disclosed
WO-2009112475-A1 PYRROLO [2, 3-B] PYRIDIN DERIVATIVES AS IKK2 INHIBITORS GLAXO GROUP LIMITED (GB) 2009-09-17 WO disclosed