SCHEMBL4060742

SCHEMBL4060742

COc1ccc(C2(C#N)CCc3ncncc3C2)c2c3ccccc3n(C)c12

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
ALOX15 P16050 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
GABRP O00591 1/20 0.32
GABRD O14764 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRB1 P18505 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32
GABRA3 P34903 1/20 0.32
GABRA2 P47869 1/20 0.32
GABRB2 P47870 1/20 0.32
GABRA4 P48169 1/20 0.32
GABRE P78334 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4540659 0.89 KDM4E (0.32) KDM4EHDAC9
SCHEMBL4054950 0.87 KDM4E (0.32) HSD17B10GABRPGABRDGABRA1GABRB1
SCHEMBL4053327 0.84 CYP17A1 (0.37) HSD17B10CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL4062215 0.84 KDR (0.34) HSD17B10TP53MAPTKDRMYLK
SCHEMBL4051543 0.83 KDR (0.32) TP53MAPTKDRMYLKKDM4E
SCHEMBL4059118 0.81 CYP17A1 (0.35)
SCHEMBL4018297 0.81 CYP17A1 (0.33) HSD17B10MAPTKDM4EALDH1A1HPGD
SCHEMBL13693694 0.78 PDE4A (0.41) HSD17B10TP53KDRMYLKKDM4E
SCHEMBL4233727 0.78 KDR (0.30) KDRMYLK
SCHEMBL4052813 0.76 KDM4E (0.31) HSD17B10KDM4EALDH1A1GLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO claimed
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed