SCHEMBL4065119

SCHEMBL4065119

CCS(=O)(=O)Nc1ccc2c(c1)S(=O)(=O)C=C(c1c(O)c3cc(F)ccc3n(CCC3CC3)c1=O)N2

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.54
NR1I2 O75469 1/20 0.54
PLK1 P53350 2/20 0.35
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
PARG Q86W56 1/20 0.33
BRD4 O60885 9/20 0.33
HTR2A P28223 1/20 0.32
DRD3 P35462 1/20 0.32
CRY1 Q16526 2/20 0.32
CRY2 Q49AN0 2/20 0.32
BRD2 P25440 1/20 0.32
ADORA2B P29275 1/20 0.32
TSPO P30536 1/20 0.32
EP300 Q09472 1/20 0.32
BRD3 Q15059 1/20 0.32
BRDT Q58F21 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4072462 0.95 CYP2C9 (0.52) CYP2C9NR1I2PLK1PARGBRD4
SCHEMBL3921871 0.93 CYP2C9 (0.55) CYP2C9NR1I2PLK1CNR1CNR2
SCHEMBL3921480 0.92 CYP2C9 (0.55) CYP2C9NR1I2PLK1PARGBRD4
SCHEMBL4065684 0.91 CYP2C9 (0.54) CYP2C9NR1I2PLK1PARGBRD4
SCHEMBL3924684 0.89 CYP2C9 (0.56) CYP2C9NR1I2PARGBRD4
SCHEMBL4068112 0.87 CYP2C9 (0.39) CYP2C9NR1I2PARGBRD4
SCHEMBL3929718 0.87 CYP2C9 (0.54) CYP2C9NR1I2PLK1CRY1CRY2
SCHEMBL4067186 0.86 CYP2C9 (0.49) CYP2C9NR1I2PLK1PARG
SCHEMBL3922170 0.84 CYP2C9 (0.54) CYP2C9NR1I2PLK1CRY1CRY2
SCHEMBL3921287 0.84 CYP2C9 (0.72) CYP2C9NR1I2PLK1CRY1CRY2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1786807-B1 HETEROCYCLIC ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2009-07-29 EP claimed