SCHEMBL4065656

SCHEMBL4065656

Cc1[nH]c2c(F)ccc(C)c2c1CCNc1ncnc2cc(-c3ccc(-c4ccccc4)cc3)sc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT1 P17948 9/20 0.45
EGFR P00533 8/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
TYK2 P29597 1/20 0.44
KDR P35968 2/20 0.43
PRKCI P41743 1/20 0.38
IKBKB O14920 2/20 0.38
CHUK O15111 1/20 0.36
POLB P06746 1/20 0.36
RAD52 P43351 1/20 0.36
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35
TUBA4A P68366 1/20 0.35
TUBB4B P68371 1/20 0.35
TUBB3 Q13509 1/20 0.35
TUBB2A Q13885 1/20 0.35
TUBB8 Q3ZCM7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4071195 0.98 FLT1 (0.46) FLT1EGFRNPC1RAB9ATYK2
SCHEMBL3930445 0.97 FLT1 (0.43) FLT1EGFRNPC1RAB9ATYK2
SCHEMBL3937751 0.93 NPC1 (0.46) FLT1EGFRNPC1RAB9ATYK2
SCHEMBL4068409 0.93 TYK2 (0.53) FLT1EGFRNPC1RAB9ATYK2
SCHEMBL4069302 0.92 NPC1 (0.44) FLT1EGFRNPC1RAB9ATYK2
SCHEMBL3930923 0.92 NPC1 (0.42) FLT1EGFRNPC1RAB9ATYK2
SCHEMBL3939022 0.92 NPC1 (0.45) FLT1EGFRNPC1RAB9ATYK2
SCHEMBL4073363 0.91 NPC1 (0.43) FLT1EGFRNPC1RAB9ATYK2
SCHEMBL3936128 0.91 NPC1 (0.43) FLT1EGFRNPC1RAB9ATYK2
SCHEMBL4067376 0.91 FLT1 (0.48) FLT1EGFRNPC1RAB9ATYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090042913-A1 Indolylalkylthienopyrimidylamines as modulators of the EP2 receptor BAYER SCHERING PHARMA AG (DE) 2009-02-12 US claimed
EP-2014662-A1 Indolyl alkyl thieno-pyrimidyl amines as modulators of EP2 receptors Bayer Schering Pharma Aktiengesellschaft (DE) 2009-01-14 EP claimed
US-20090042913-A1 Indolylalkylthienopyrimidylamines as modulators of the EP2 receptor BAYER SCHERING PHARMA AG (DE) 2009-02-12 US disclosed
US-20090042913-A1 Indolylalkylthienopyrimidylamines as modulators of the EP2 receptor BAYER SCHERING PHARMA AG (DE) 2009-02-12 US disclosed
US-20090042913-A1 Indolylalkylthienopyrimidylamines as modulators of the EP2 receptor BAYER SCHERING PHARMA AG (DE) 2009-02-12 US disclosed
EP-2014662-A1 Indolyl alkyl thieno-pyrimidyl amines as modulators of EP2 receptors Bayer Schering Pharma Aktiengesellschaft (DE) 2009-01-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090042913-A1 Indolylalkylthienopyrimidylamines as modulators of the EP2 receptor PTGER2, PTGER1, PTGDR2 FLT1 3775/4885EGFR 498/4885NPC1 2246/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.