SCHEMBL4065766

SCHEMBL4065766

Cc1ncnc(C)c1OC(=O)NCc1ccc(CN(C2CCNCC2)C2CCCc3cccnc32)cc1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 16/20 0.40
CYP2D6 P10635 15/20 0.40
CYP3A4 P08684 9/20 0.40
HDAC1 Q13547 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4061006 0.93 CXCR4 (0.41) CXCR4CYP2D6CYP3A4
SCHEMBL4070057 0.92 CXCR4 (0.39) CXCR4CYP2D6CYP3A4
SCHEMBL4066923 0.88 CXCR4 (0.41) CXCR4CYP2D6CYP3A4HDAC1HDAC6
SCHEMBL4061365 0.83 HDAC1 (0.40) CXCR4CYP2D6CYP3A4HDAC1HDAC6
SCHEMBL4072439 0.82 CXCR4 (0.47) CXCR4CYP2D6CYP3A4
SCHEMBL4065284 0.81 CXCR4 (0.42) CXCR4CYP2D6CYP3A4
SCHEMBL4063233 0.81 CXCR4 (0.45) CXCR4CYP2D6CYP3A4
SCHEMBL4065894 0.81 CXCR4 (0.44) CXCR4CYP2D6CYP3A4
SCHEMBL4060854 0.81 CXCR4 (0.43) CXCR4CYP2D6CYP3A4
SCHEMBL4064523 0.80 CXCR4 (0.42) CXCR4CYP2D6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317443-B1 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS ANORMED INC (CA) 2009-01-14 EP claimed