SCHEMBL4068673

SCHEMBL4068673

Cc1ncnc(C)c1OC(=O)NCc1cccc(CN(Cc2ncco2)C2CCCc3cccnc32)c1

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 18/20 0.42
CYP2D6 P10635 9/20 0.42
CYP3A4 P08684 7/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4070871 0.94 CXCR4 (0.44) CXCR4CYP2D6CYP3A4
SCHEMBL4064271 0.94 CXCR4 (0.42) CXCR4CYP2D6CYP3A4
SCHEMBL4062065 0.93 CXCR4 (0.44) CXCR4CYP2D6CYP3A4
SCHEMBL4066865 0.89 CXCR4 (0.43) CXCR4CYP2D6CYP3A4
SCHEMBL4071653 0.88 CXCR4 (0.41) CXCR4CYP2D6CYP3A4
SCHEMBL4068095 0.88 CXCR4 (0.42) CXCR4CYP2D6CYP3A4
SCHEMBL4064243 0.87 CXCR4 (0.47) CXCR4CYP2D6CYP3A4
SCHEMBL4071779 0.86 CXCR4 (0.42) CXCR4CYP2D6CYP3A4
SCHEMBL4068777 0.86 CXCR4 (0.43) CXCR4CYP2D6CYP3A4
SCHEMBL4061217 0.86 CXCR4 (0.44) CXCR4CYP2D6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317443-B1 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS ANORMED INC (CA) 2009-01-14 EP claimed