SCHEMBL4069559

SCHEMBL4069559

CCc1c(C(N)=O)cccc1C(F)CC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.40
RPS6KB1 P23443 3/20 0.36
CXCR2 P25025 1/20 0.35
IRAK4 Q9NWZ3 1/20 0.35
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 3/20 0.34
MAPT P10636 2/20 0.34
HPGD P15428 2/20 0.34
HSD17B10 Q99714 2/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 2/20 0.34
LMNA P02545 2/20 0.34
MEN1 O00255 1/20 0.34
NR1I2 O75469 1/20 0.34
CHRM2 P08172 1/20 0.34
CYP3A4 P08684 1/20 0.34
ADRA2A P08913 1/20 0.34
OPRK1 P41145 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4951728 0.84 PARP1 (0.42) PARP1RPS6KB1CXCR2IRAK4KEAP1
SCHEMBL45719 0.79 PARP1 (0.51) PARP1IRAK4KEAP1NFE2L2KDM4E
SCHEMBL72113 0.76 PARP1 (0.49) PARP1IRAK4KEAP1NFE2L2KDM4E
SCHEMBL8898159 0.76 CYP3A4 (0.42) PARP1RPS6KB1ALDH1A1MAPTTSHR
SCHEMBL30499962 0.75 MAPK8 (0.47) PARP1KDM4EALDH1A1MAPTHPGD
SCHEMBL19695740 0.75 MAPK8 (0.47) PARP1KDM4EALDH1A1MAPTHPGD
SCHEMBL17182410 0.75 KDM4E (0.40) PARP1RPS6KB1CXCR2KDM4EALDH1A1
Charcoal, Activated SCHEMBL9345241 0.74 PARP1 (0.47) PARP1IRAK4KEAP1NFE2L2KDM4E
SCHEMBL6321332 0.74 PARP1 (0.47) PARP1IRAK4KEAP1NFE2L2KDM4E
Hydrochloric Acid SCHEMBL7467552 0.74 PARP1 (0.47) PARP1IRAK4KEAP1NFE2L2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2040555-A2 FORMULATED TICK AND INSECT REPELLENT COMPOSITIONS E.I. DU PONT DE NEMOURS AND COMPANY (US) 2009-04-01 EP disclosed
WO-2007133683-A2 FORMULATED TICK AND INSECT REPELLENT COMPOSITIONS E. I. DU PONT DE NEMOURS AND COMPANY (US) 2007-11-22 WO disclosed