SCHEMBL40698

SCHEMBL40698

CCCc1cnc2cc(Cl)ccc2c1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 2/20 0.47
PDGFRA P16234 2/20 0.47
NR4A2 P43354 1/20 0.43
MAOB P27338 4/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
PDE10A Q9Y233 4/20 0.41
HRH4 Q9H3N8 2/20 0.39
DAO P14920 1/20 0.39
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
TRPV1 Q8NER1 1/20 0.36
RAB9A P51151 1/20 0.36
TEC P42680 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12507578 0.86 PDGFRB (0.50) PDGFRBPDGFRANR4A2MAOBKMT2A
SCHEMBL26323741 0.84 PDGFRB (0.45) PDGFRBPDGFRAMAOBPDE10ATRPV1
SCHEMBL16880666 0.81 PDGFRB (0.51) PDGFRBPDGFRANR4A2MAOBKMT2A
SCHEMBL28169400 0.79 PDGFRB (0.50) PDGFRBPDGFRANR4A2MAOBKMT2A
SCHEMBL16891547 0.79 PDGFRB (0.50) PDGFRBPDGFRANR4A2MAOBKMT2A
SCHEMBL17785411 0.79 PDGFRB (0.50) PDGFRBPDGFRANR4A2MAOBKMT2A
SCHEMBL6115113 0.77 TRPV1 (0.55) PDGFRBPDGFRAMAOBKMT2AMEN1
Ammonia Solution, Strong SCHEMBL5507007 0.76 TRPV1 (0.53) PDGFRBPDGFRAMAOBKMT2AMEN1
SCHEMBL29115356 0.75 NPC1 (0.52) PDGFRBPDGFRAKMT2AMEN1CYP1A2
SCHEMBL24447290 0.75 KDM4C (0.41) PDGFRBPDGFRAPDE10ATRPV1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3154343-A1 USE AS RODENTICIDES OF COMPOUNDS THAT INHIBIT BLOOD COAGULATION Gulba, Dietrich (DE) 2017-04-19 EP disclosed
WO-2015189331-A1 USE AS RODENTICIDES OF COMPOUNDS THAT INHIBIT BLOOD COAGULATION GULBA DIETRICH (DE) 2015-12-17 WO disclosed
EP-2422194-A1 VESICULAR SYSTEM AND USES THEREOF Agency For Science, Technology And Research (SG) 2012-02-29 EP disclosed
WO-2012008916-A1 FLAME RETARDANT AND INTUMESCENT COMPOUND AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2012-01-19 WO disclosed
WO-2012002913-A1 PROCESS OF FORMING A CYCLIC IMIDE NANYANG TECHNOLOGICAL UNIVERSITY (SG) 2012-01-05 WO disclosed
WO-2011034506-A1 PROCESS OF FORMING AN AMIDE NANYANG TECHNOLOGICAL UNIVERSITY (SG) 2011-03-24 WO disclosed
WO-2010132029-A1 OCTAHYDRO BIQUINOLINE COMPOUND NANYANG TECHNOLOGICAL UNIVERSITY (SG) 2010-11-18 WO disclosed
WO-2010123462-A1 VESICULAR SYSTEM AND USES THEREOF AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2010-10-28 WO disclosed
WO-2010090596-A1 HOLLOW SILICA PARTICLE WITH A POLYMER THEREON AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2010-08-12 WO disclosed
WO-2010044752-A1 AMPHIPHILIC POLYMERS AND NANOCRYSTALS COATED THEREWITH AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2010-04-22 WO disclosed
WO-2010027326-A1 PEPTIDE NUCLEIC ACID MONOMERS AND OLIGOMERS NANYANG TECHNOLOGICAL UNIVERSITY (SG) 2010-03-11 WO disclosed
WO-2009142604-A1 POLYMER ENCAPSULATED PARTICLES AS SURFACE ENHANCED RAMAN SCATTERING PROBES NANYANG TECHNOLOGICAL UNIVERSITY (SG) 2009-11-26 WO disclosed
EP-2084105-A1 METHOD OF FUNCTIONALIZING A CARBON MATERIAL Agency for Science, Technology And Research (SG) 2009-08-05 EP disclosed
WO-2009078813-A1 METHOD OF FORMING OSELTAMIVIR AND DERIVATIVES THEREOF NANYANG TECHNOLOGICAL UNIVERSITY (SG) 2009-06-25 WO disclosed
WO-2009038544-A1 AMPHIPHILIC POLYMER AND PROCESSES OF FORMING THE SAME AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2009-03-26 WO disclosed
WO-2009029053-A1 METHOD OF COATING A PARTICLE AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2009-03-05 WO disclosed
WO-2008048192-A1 METHOD OF FUNCTIONALIZING A CARBON MATERIAL AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH (SG) 2008-04-24 WO disclosed
WO-2007097719-A1 CYCLISATION PROCESS OF FORMING A MULTIPLE RING COMPOUND NANYANG TECHNOLOGICAL UNIVERSITY (SG) 2007-08-30 WO disclosed