SCHEMBL4070879

SCHEMBL4070879

N[C@H]1CN(C(=O)O)c2ccccc2N(CCOCc2ccccc2)C1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TEAD3 Q99594 2/20 0.38
LTA4H P09960 1/20 0.36
CYP3A4 P08684 2/20 0.36
XIAP P98170 2/20 0.36
CYP2C19 P33261 1/20 0.36
CCKBR P32239 3/20 0.36
ACE P12821 1/20 0.35
GBA1 P04062 2/20 0.35
UGCG Q16739 2/20 0.35
GBA2 Q9HCG7 2/20 0.35
SLC6A1 P30531 2/20 0.35
AGTR2 P50052 1/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4251386 0.89 GAA (0.40) GAAMEN1KMT2ATEAD3LTA4H
Hydrochloric Acid SCHEMBL4251381 0.88 GAA (0.39) GAAMEN1KMT2ATEAD3CYP3A4
Hydrochloric Acid SCHEMBL4993066 0.88 GAA (0.39) GAAMEN1KMT2ATEAD3CYP3A4
SCHEMBL14093724 0.85 GAA (0.39) GAAMEN1KMT2ATEAD3CYP3A4
SCHEMBL4988616 0.85 GAA (0.39) GAAMEN1KMT2ATEAD3CYP3A4
Hydrochloric Acid SCHEMBL4988622 0.84 GAA (0.38) GAAMEN1KMT2ATEAD3CYP3A4
Hydrochloric Acid SCHEMBL4988609 0.84 GAA (0.38) GAAMEN1KMT2ATEAD3CYP3A4
SCHEMBL8213549 0.80 NPC1 (0.34) GAAMEN1KMT2ATEAD3CYP3A4
SCHEMBL8209635 0.79 GAA (0.36) GAAMEN1KMT2ATEAD3LTA4H
Hydrochloric Acid SCHEMBL4993551 0.78 GAA (0.35) GAAMEN1KMT2ATEAD3LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2069317-A2 4-OXO-2,3,4,5-TETRAHYDRO-BENZO[B][1,4]DIAZEPINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-06-17 EP disclosed
WO-2008034735-A2 4-OXO-2,3,4,5-TETRAHYDRO-BENZO[B][1,4]DIAZEPINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-03-27 WO disclosed