SCHEMBL4073091

SCHEMBL4073091

CC(C)=CCn1c([C@H]2CCC[C@@H](N)C2)nc2c1c(=O)n(C)c(=O)n2C

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 14/20 0.62
KMT2A Q03164 2/20 0.48
LMNA P02545 1/20 0.48
MAPK1 P28482 1/20 0.48
ADORA2A P29274 2/20 0.48
ADORA2B P29275 2/20 0.48
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
CHRM1 P11229 2/20 0.46
CHRM2 P08172 1/20 0.46
CHRM3 P20309 1/20 0.46
KCNH2 Q12809 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL555408 1.00 DPP4 (0.62) DPP4KMT2ALMNAMAPK1ADORA2A
SCHEMBL4073092 1.00 DPP4 (0.62) DPP4KMT2ALMNAMAPK1ADORA2A
Hydrochloric Acid SCHEMBL555194 0.99 DPP4 (0.61) DPP4KMT2ALMNAMAPK1ADORA2A
Hydrochloric Acid SCHEMBL27582646 0.99 DPP4 (0.61) DPP4KMT2ALMNAMAPK1ADORA2A
Hydrochloric Acid SCHEMBL555193 0.99 DPP4 (0.61) DPP4KMT2ALMNAMAPK1ADORA2A
SCHEMBL556432 0.94 DPP4 (0.59) DPP4KMT2ALMNAMAPK1ADORA2A
SCHEMBL556285 0.87 DPP4 (0.61) DPP4KMT2ALMNAMAPK1ADORA2A
SCHEMBL557054 0.87 DPP4 (0.52) DPP4KMT2ALMNAMAPK1ADORA2A
SCHEMBL556313 0.86 DPP4 (0.51) DPP4KMT2ALMNAMAPK1ADORA2A
SCHEMBL556304 0.85 DPP4 (0.50) DPP4KMT2ALMNAMAPK1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2298769-B1 Xanthin derivatives, their production and utilisation as medicine BOEHRINGER INGELHEIM PHARMA (DE) 2013-10-30 EP claimed
EP-1757606-B1 Xanthinderivatives for use as medical agents and the preparation thereof BOEHRINGER INGELHEIM PHARMA (DE) 2009-05-06 EP claimed
EP-1368349-B1 XANTHINE DERIVATIVE, PRODUCTION AND USE THEREOF AS A MEDICAMENT BOEHRINGER INGELHEIM PHARMA (DE) 2007-02-14 EP claimed