SCHEMBL4074050

SCHEMBL4074050

Nc1ccccc1NC(=O)c1ccc(N2CCCC3(CCN(C(=O)O)C3)C2)nc1

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 20/20 0.67
KCNH2 Q12809 8/20 0.67
HDAC3 O15379 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4067024 0.96 HDAC1 (0.70) HDAC1KCNH2HDAC3
SCHEMBL4069251 0.95 HDAC1 (0.73) HDAC1KCNH2HDAC3
SCHEMBL4073227 0.92 HDAC1 (0.70) HDAC1KCNH2HDAC3
SCHEMBL4070242 0.91 HDAC1 (0.71) HDAC1KCNH2HDAC3
SCHEMBL4068946 0.91 HDAC1 (0.70) HDAC1KCNH2HDAC3
SCHEMBL4072390 0.90 HDAC1 (0.70) HDAC1KCNH2HDAC3
SCHEMBL1639270 0.90 HDAC1 (0.71) HDAC1KCNH2HDAC3
SCHEMBL1640945 0.88 HDAC1 (0.71) HDAC1KCNH2HDAC3
SCHEMBL1640642 0.88 HDAC1 (0.72) HDAC1KCNH2HDAC3
SCHEMBL4069836 0.87 HDAC1 (0.72) HDAC1KCNH2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1954698-B1 SPIROCYCLIC COMPOUNDS AS HDAC INHIBITORS MERCK & CO INC (US) 2009-06-24 EP claimed