SCHEMBL4074747

SCHEMBL4074747

COc1cc([C]c2ccc(F)c(F)c2)ccc1CN1CCC2(CC1)OCc1ccncc12

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 12/20 0.44
MCHR1 Q99705 10/20 0.44
MELK Q14680 1/20 0.37
OPRM1 P35372 2/20 0.36
OPRK1 P41145 1/20 0.36
AVPR1A P37288 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4074742 1.00 KCNH2 (0.44) KCNH2MCHR1MELKOPRM1OPRK1
SCHEMBL4074749 0.87 MCHR1 (0.49) KCNH2MCHR1
SCHEMBL13664939 0.85 MCHR1 (0.57) KCNH2MCHR1AVPR1A
SCHEMBL4076927 0.80 MCHR1 (0.53) KCNH2MCHR1AVPR1A
SCHEMBL4076908 0.80 MCHR1 (0.53) KCNH2MCHR1AVPR1A
SCHEMBL4076904 0.80 MCHR1 (0.53) KCNH2MCHR1AVPR1A
SCHEMBL13664942 0.76 MCHR1 (0.64) KCNH2MCHR1AVPR1A
SCHEMBL4076079 0.76 MCHR1 (0.64) KCNH2MCHR1OPRM1OPRK1AVPR1A
SCHEMBL4252556 0.76 MCHR1 (0.64) KCNH2MCHR1OPRM1OPRK1AVPR1A
SCHEMBL13664934 0.75 MCHR1 (0.60) KCNH2MCHR1OPRM1AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2072519-A1 DIARYL KETIMINE DERIVATIVE BANYU PHARMACEUTICAL CO., LTD. (JP) 2009-06-24 EP disclosed