SCHEMBL4075363

SCHEMBL4075363

O=c1ccc2cnc(Nc3ccncc3)nc2[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 5/20 0.50
CCND1 P24385 5/20 0.50
CCND2 P30279 5/20 0.50
CCND3 P30281 5/20 0.50
PDE3B Q13370 2/20 0.46
PDE3A Q14432 2/20 0.46
MAPK8 P45983 1/20 0.41
MAPK9 P45984 1/20 0.41
MAPK10 P53779 1/20 0.41
PIK3C3 Q8NEB9 1/20 0.41
FGFR1 P11362 3/20 0.40
EGFR P00533 2/20 0.40
SRC P12931 2/20 0.40
JAK1 P23458 1/20 0.40
TYK2 P29597 1/20 0.40
CCNA2 P20248 3/20 0.39
CDK2 P24941 3/20 0.39
BRAF P15056 1/20 0.38
CAMK2D Q13557 1/20 0.38
CCNB2 O95067 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5264282 0.86 CDK4 (0.52) CDK4CCND1CCND2CCND3MAPK8
SCHEMBL2320862 0.85 EGFR (0.43) CDK4CCND1CCND2CCND3PDE3B
SCHEMBL748173 0.77 CCND3 (0.49) CDK4CCND1CCND2CCND3MAPK8
SCHEMBL29979953 0.76 JAK1 (0.50) JAK1TYK2
SCHEMBL16416249 0.76 MAPK8 (0.48) PDE3BPDE3AMAPK8MAPK9MAPK10
SCHEMBL10346428 0.74 CDK4 (0.61) CDK4CCND1CCND2CCND3FGFR1
SCHEMBL20400864 0.73 SYK (0.51) CDK4CCND1CCND2CCND3MAPK8
SCHEMBL30950984 0.72 BRAF (0.46) PDE3BPDE3AMAPK8MAPK9MAPK10
SCHEMBL16993339 0.72 CDK4 (0.51) CDK4CCND1CCND2CCND3PDE3B
SCHEMBL17910166 0.72 MAPK8 (0.54) CDK4CCND1CCND2CCND3PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1751155-B1 SUBSTITUTED AZACHINAZOLINES HAVING AN ANTIVIRAL ACTION BAYER HEALTHCARE AG (DE) 2009-01-07 EP disclosed