SCHEMBL4076276

SCHEMBL4076276

Clc1ccc(Cl)c(CC2(NNC3(Cc4cccc(Cl)c4Cl)CCN(c4ncnc5[nH]ccc45)CC3)CCN(c3ncnc4[nH]ccc34)CC2)c1

nearest known ligand 0.69

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AKT2 P31751 19/20 0.69
AKT1 P31749 4/20 0.59
GSK3B P49841 4/20 0.53
RPS6KB1 P23443 2/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4076275 0.90 AKT2 (0.86) AKT2AKT1GSK3BRPS6KB1CYP2D6
SCHEMBL1003955 0.82 AKT2 (1.00) AKT2AKT1GSK3BRPS6KB1CYP2D6
SCHEMBL1001810 0.82 AKT2 (1.00) AKT2AKT1GSK3BRPS6KB1CYP2D6
SCHEMBL3993935 0.81 AKT2 (0.76) AKT2AKT1GSK3BRPS6KB1CYP2D6
SCHEMBL3917909 0.79 AKT2 (0.61) AKT2AKT1GSK3BRPS6KB1CYP2D6
SCHEMBL1001877 0.76 AKT2 (1.00) AKT2AKT1GSK3BRPS6KB1CYP2D6
SCHEMBL1003441 0.75 AKT2 (1.00) AKT2AKT1GSK3BRPS6KB1CYP2D6
SCHEMBL3930367 0.73 AKT2 (0.68) AKT2AKT1GSK3BRPS6KB1CYP2D6
SCHEMBL3917914 0.73 AKT2 (0.70) AKT2AKT1GSK3BRPS6KB1CYP2D6
SCHEMBL1002688 0.73 AKT2 (1.00) AKT2AKT1GSK3BRPS6KB1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2037931-A2 PHARMACEUTICAL COMBINATIONS OF PK INHIBITORS AND OTHER ACTIVE AGENTS Astex Therapeutics Limited (GB) 2009-03-25 EP disclosed
WO-2007125310-A2 PHARMACEUTICAL COMBINATIONS OF PK INHIBITORS AND OTHER ACTIVE AGENTS ASTEX THERAPEUTICS LIMITED (GB) 2007-11-08 WO disclosed