SCHEMBL4086192

SCHEMBL4086192

O=C(O)Cc1ccccc1CCBr

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.57
TDP1 Q9NUW8 2/20 0.50
BCAT2 O15382 1/20 0.44
PTPN1 P18031 1/20 0.43
GSK3B P49841 1/20 0.43
CXCL8 P10145 5/20 0.43
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.43
MAPT P10636 1/20 0.43
PTGS2 P35354 2/20 0.41
PTGS1 P23219 2/20 0.41
AKR1B10 O60218 1/20 0.41
UGT1A9 O60656 1/20 0.41
TRPA1 O75762 1/20 0.41
ABCB11 O95342 1/20 0.41
MT-CO2 P00403 1/20 0.41
TTR P02766 1/20 0.41
ALB P02768 1/20 0.41
UGT1A6 P19224 1/20 0.41
UGT1A1 P22309 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11548652 0.88 AKR1B1 (0.53) AKR1B1TDP1BCAT2CXCL8KDM4E
SCHEMBL30359 0.84 AKR1B1 (0.76) AKR1B1TDP1BCAT2CXCL8KDM4E
SCHEMBL29410826 0.84 AKR1B1 (0.76) AKR1B1TDP1BCAT2CXCL8KDM4E
SCHEMBL76036 0.83 AKR1B1 (0.61) AKR1B1TDP1BCAT2CXCL8KDM4E
SCHEMBL28842838 0.82 AKR1B1 (0.73) AKR1B1TDP1BCAT2CXCL8KDM4E
Hydrogen Sulfide SCHEMBL27426416 0.82 AKR1B1 (0.73) AKR1B1TDP1BCAT2CXCL8KDM4E
Hydrochloric Acid SCHEMBL9621764 0.82 AKR1B1 (0.73) AKR1B1TDP1BCAT2CXCL8KDM4E
Hydrochloric Acid SCHEMBL6767821 0.82 AKR1B1 (0.73) AKR1B1TDP1BCAT2CXCL8KDM4E
Iodide SCHEMBL31305035 0.82 AKR1B1 (0.73) AKR1B1TDP1BCAT2CXCL8KDM4E
SCHEMBL3124446 0.81 AKR1B1 (0.59) AKR1B1TDP1BCAT2PTPN1CXCL8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7488748-B2 3,6-Disubstituted azabicyclo hexane derivatives as muscarinic receptor antagonists RANBAXY LABORATORIES LIMITED (IN) 2009-02-10 US disclosed
US-20060247225-A1 3,6-Disubstituted azabicyclo hexane derivatives as muscarinic receptor antagonists RANBAXY LABORATORIES LIMITED (IN) 2006-11-02 US disclosed
EP-1590325-A1 3,6-DISUBSTITUTED AZABICYCLO HEXANE DERIVATIVES AS MUSCARINIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES, LTD. (IN) 2005-11-02 EP disclosed
WO-2004067510-A1 3,6-DISUBSTITUTED AZABICYCLO HEXANE DERIVATIVES AS MUSCARINIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2004-08-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060247225-A1 3,6-Disubstituted azabicyclo hexane derivatives as muscarinic receptor antagonists CHRM3, CHRM5, CHRM2 AKR1B1 436/4885TDP1 4627/4885BCAT2 4313/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.