SCHEMBL4087664

SCHEMBL4087664

Cc1ccc(NC(=O)c2ccc(C=CC(=O)NOC3CCCCO3)s2)cc1Nc1nc(-c2cccnc2)cs1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 16/20 0.56
PDGFRB P09619 7/20 0.56
HDAC3 O15379 6/20 0.56
KDR P35968 6/20 0.56
HDAC4 P56524 6/20 0.56
HDAC1 Q13547 6/20 0.56
HDAC7 Q8WUI4 6/20 0.56
HDAC2 Q92769 6/20 0.56
HDAC10 Q969S8 6/20 0.56
HDAC11 Q96DB2 6/20 0.56
HDAC8 Q9BY41 6/20 0.56
HDAC6 Q9UBN7 6/20 0.56
HDAC9 Q9UKV0 6/20 0.56
HDAC5 Q9UQL6 6/20 0.56
BCR P11274 11/20 0.55
KIT P10721 2/20 0.48
EGFR P00533 1/20 0.48
ERBB2 P04626 1/20 0.48
LCK P06239 1/20 0.48
FYN P06241 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4087660 1.00 ABL1 (0.56) ABL1PDGFRBHDAC3KDRHDAC4
SCHEMBL6531698 0.91 ABL1 (0.51) ABL1PDGFRBHDAC3KDRHDAC4
SCHEMBL4080309 0.91 ABL1 (0.54) ABL1PDGFRBHDAC3KDRHDAC4
SCHEMBL4080315 0.91 ABL1 (0.54) ABL1PDGFRBHDAC3KDRHDAC4
SCHEMBL4079765 0.89 ABL1 (0.72) ABL1PDGFRBHDAC3KDRHDAC4
SCHEMBL4079758 0.89 ABL1 (0.72) ABL1PDGFRBHDAC3KDRHDAC4
Water SCHEMBL4087659 0.84 ABL1 (0.60) ABL1PDGFRBHDAC3KDRHDAC4
SCHEMBL4082784 0.84 ABL1 (0.78) ABL1PDGFRBHDAC3KDRHDAC4
SCHEMBL4082778 0.84 ABL1 (0.78) ABL1PDGFRBHDAC3KDRHDAC4
SCHEMBL4079841 0.79 ABL1 (0.56) ABL1PDGFRBHDAC3KDRHDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2060565-A1 Novel bifunctional compounds which inhibit protein kinases and histone deacetylases 4SC AG (DE) 2009-05-20 EP disclosed