SCHEMBL4087988

SCHEMBL4087988

Cc1cc2c(nc1C)[nH]c1c(C(=O)NCCN3CCCC3)cccc12

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
POLR1A O95602 10/20 0.55
SMYD2 Q9NRG4 3/20 0.47
PARP1 P09874 1/20 0.46
KDM4E B2RXH2 1/20 0.45
HSD17B10 Q99714 1/20 0.45
PDK2 Q15119 1/20 0.45
KCNH2 Q12809 1/20 0.44
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4087694 0.79 PDK2 (0.50) POLR1AKDM4EHSD17B10PDK2KCNH2
SCHEMBL3890307 0.74 PDK2 (0.50) PARP1KDM4EHSD17B10PDK2KCNH2
SCHEMBL14430692 0.73 KMT2A (0.61) SMYD2PARP1KDM4EHSD17B10KCNH2
SCHEMBL13164061 0.73 NPSR1 (0.59) POLR1ANPSR1
SCHEMBL28598516 0.72 NPSR1 (0.56) POLR1ASMYD2KCNH2NPSR1
SCHEMBL13164063 0.72 NPSR1 (0.58) POLR1AKDM4EHSD17B10NPSR1
SCHEMBL25970713 0.71 POLR1A (1.00) POLR1AKCNH2
SCHEMBL18760971 0.69 NPSR1 (0.54) POLR1ANPSR1
SCHEMBL10803261 0.69 SMYD2 (0.54) POLR1ASMYD2PARP1KDM4ENPSR1
SCHEMBL25346201 0.69 POLR1A (0.76) POLR1AHSD17B10KCNH2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079696-A2 KINASE INHIBITORS Takeda San Diego, Inc. (US) 2009-07-22 EP disclosed
WO-2008054956-A2 KINASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2008-05-08 WO disclosed