SCHEMBL411237

SCHEMBL411237

CCN(CC(NC(=O)Cn1nc(-c2ccc(Cl)cc2)n(C[C@H](O)C(F)(F)F)c1=O)c1cccc(C(F)(F)F)c1)C(=O)O

nearest known ligand 0.68

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 20/20 0.68
AVPR1A P37288 20/20 0.68
SLC6A2 P23975 1/20 0.45
OXTR P30559 1/20 0.45
OPRK1 P41145 1/20 0.45
AVPR1B P47901 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL411180 0.91 AVPR2 (0.70) AVPR2AVPR1ASLC6A2OXTROPRK1
SCHEMBL16673951 0.90 AVPR2 (0.74) AVPR2AVPR1ASLC6A2OXTROPRK1
SCHEMBL419513 0.87 AVPR2 (0.77) AVPR2AVPR1A
SCHEMBL408829 0.87 AVPR2 (0.81) AVPR2AVPR1A
SCHEMBL10217399 0.87 AVPR2 (0.76) AVPR2AVPR1A
SCHEMBL19244822 0.86 AVPR2 (0.66) AVPR2AVPR1A
SCHEMBL3447408 0.86 AVPR2 (0.75) AVPR2AVPR1A
Hydrochloric Acid SCHEMBL3446983 0.86 AVPR2 (0.75) AVPR2AVPR1A
SCHEMBL19265141 0.86 AVPR2 (0.75) AVPR2AVPR1A
SCHEMBL413603 0.85 AVPR2 (0.72) AVPR2AVPR1ASLC6A2OXTROPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408751-A1 Substituted 2-acetamido-5-aryl-1,2,4-triazolones and use thereof Bayer Pharma Aktiengesellschaft (DE) 2012-01-25 EP disclosed
WO-2010105770-A1 SUBSTITUTED 2-ACETAMIDO-5-ARYL-1,2,4-TRIAZOLONES AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-09-23 WO disclosed