SCHEMBL4119281

SCHEMBL4119281

O=C(O)NC1CCC(CN2CCCCC2)CC1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.52
ADRA2C P18825 1/20 0.52
CCR1 P32246 4/20 0.47
SMN1; SMN2 Q16637 1/20 0.45
MAPT P10636 3/20 0.45
ALDH1A1 P00352 1/20 0.44
MAPK1 P28482 1/20 0.44
CHRM2 P08172 4/20 0.43
CHRM1 P11229 4/20 0.43
CHRM3 P20309 4/20 0.43
FPR3 P25089 1/20 0.43
FPR2 P25090 1/20 0.43
TP53 P04637 1/20 0.42
GAA P10253 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4119272 1.00 CHRM5 (0.52) CHRM5ADRA2CCCR1SMN1; SMN2MAPT
SCHEMBL15191011 0.98 CHRM5 (0.48) CHRM5ADRA2CCCR1SMN1; SMN2MAPT
SCHEMBL15130431 0.98 CHRM5 (0.48) CHRM5ADRA2CCCR1SMN1; SMN2MAPT
SCHEMBL4909423 0.87 CCR1 (0.50) CCR1SMN1; SMN2CHRM2CHRM1CHRM3
SCHEMBL5555057 0.86 CCR1 (0.60) CHRM5ADRA2CCCR1SMN1; SMN2CHRM2
SCHEMBL27232352 0.83 CHRM3 (0.49) CHRM5CCR1CHRM2CHRM1CHRM3
SCHEMBL27224933 0.83 CHRM3 (0.49) CHRM5CCR1CHRM2CHRM1CHRM3
SCHEMBL6118868 0.83 PDE7A (0.47) CCR1SMN1; SMN2ALDH1A1GAA
SCHEMBL6118864 0.83 PDE7A (0.47) CCR1SMN1; SMN2ALDH1A1GAA
SCHEMBL27204675 0.81 KDM2B (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071519-A9 OXADIAZOLE DERIVATIVES AND THEIR USE AS NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS GLAXO GROUP LIMITED (GB) 2009-12-03 WO disclosed
WO-2009071519-A1 OXADIAZOLE DERIVATIVES AND THEIR USE AS NICOTINIC ACETYLCHOLINE RECEPTOR MODULATORS GLAXO GROUP LIMITED (GB) 2009-06-11 WO disclosed