SCHEMBL4135768

SCHEMBL4135768

COc1ncc2ccc(=O)n(CC3OCCO3)c2n1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 14/20 0.50
ALDH1A1 P00352 9/20 0.50
TSHR P16473 8/20 0.50
CYP2C19 P33261 6/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
CDK4 P11802 6/20 0.43
CCND1 P24385 6/20 0.43
CCND2 P30279 6/20 0.43
CCND3 P30281 6/20 0.43
CYP3A4 P08684 9/20 0.43
CYP2C9 P11712 4/20 0.43
HSD17B10 Q99714 6/20 0.41
HPGD P15428 4/20 0.41
USP2 O75604 2/20 0.41
CYP2D6 P10635 3/20 0.40
GLA P06280 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12090905 0.83 CDK4 (0.46) KMT2ACDK4CCND1CCND2CCND3
SCHEMBL4145936 0.81 KCNH2 (0.44) CYP1A2ALDH1A1TSHRCYP2C19MEN1
SCHEMBL4153118 0.77 CYP1A2 (0.44) CYP1A2ALDH1A1TSHRCYP2C19MEN1
SCHEMBL4136624 0.76 CDK4 (0.44) CYP1A2ALDH1A1TSHRCYP2C19CDK4
SCHEMBL12090848 0.76 KMT2A (0.42) CYP1A2ALDH1A1MEN1KMT2ACDK4
SCHEMBL19211567 0.74 CYP1A2 (0.48) CYP1A2ALDH1A1TSHRCYP2C19CDK4
SCHEMBL4149838 0.73 CDK4 (0.38) KMT2ACDK4CCND1CCND2CCND3
SCHEMBL12090780 0.73 KMT2A (0.42) CYP1A2ALDH1A1TSHRCYP2C19MEN1
SCHEMBL19211574 0.72 CDK4 (0.44) CYP1A2ALDH1A1TSHRCYP2C19CDK4
SCHEMBL19231463 0.72 CYP1A2 (0.62) CYP1A2ALDH1A1TSHRCYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2022793-B1 NOVEL HETEROCYCLIC COMPOUND OR SALT THEREOF AND INTERMEDIATE THEREOF TOYAMA CHEMICAL CO LTD (JP) 2014-06-04 EP disclosed
US-8367831-B2 Heterocyclic compound or salt thereof and intermediate thereof TOYAMA CHEMICAL CO., LTD. (JP) 2013-02-05 US disclosed
US-8367831-B2 Heterocyclic compound or salt thereof and intermediate thereof TOYAMA CHEMICAL CO., LTD. (JP) 2013-02-05 US disclosed
US-20120226035-A1 NOVEL HETEROCYCLIC COMPOUND OR SALT THEREOF AND INTERMEDIATE THEREOF TAISHO PHARMACEUTICAL CO., LTD. (JP) 2012-09-06 US disclosed
US-20120226035-A1 NOVEL HETEROCYCLIC COMPOUND OR SALT THEREOF AND INTERMEDIATE THEREOF TAISHO PHARMACEUTICAL CO., LTD. (JP) 2012-09-06 US disclosed
US-8211908-B2 Heterocyclic compound or salt thereof and intermediate thereof TOYAMA CHEMICAL CO., LTD. (JP) 2012-07-03 US disclosed
US-8211908-B2 Heterocyclic compound or salt thereof and intermediate thereof TOYAMA CHEMICAL CO., LTD. (JP) 2012-07-03 US disclosed
US-8211908-B2 Heterocyclic compound or salt thereof and intermediate thereof TOYAMA CHEMICAL CO., LTD. (JP) 2012-07-03 US disclosed
US-20090198063-A1 NOVEL HETEROCYCLIC COMPOUND OR SALT THEREOF AND INTERMEDIATE THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2009-08-06 US disclosed
US-20090198063-A1 NOVEL HETEROCYCLIC COMPOUND OR SALT THEREOF AND INTERMEDIATE THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2009-08-06 US disclosed
US-20090198063-A1 NOVEL HETEROCYCLIC COMPOUND OR SALT THEREOF AND INTERMEDIATE THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2009-08-06 US disclosed
EP-2022793-A1 NOVEL HETEROCYCLIC COMPOUND OR SALT THEREOF AND INTERMEDIATE THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2009-02-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090198063-A1 NOVEL HETEROCYCLIC COMPOUND OR SALT THEREOF AND INTERMEDIATE THEREOF IKZF3, ZC3HAV1L, H1-4 CYP1A2 1852/4885ALDH1A1 3789/4885TSHR 2873/4885
US-20120226035-A1 NOVEL HETEROCYCLIC COMPOUND OR SALT THEREOF AND INTERMEDIATE THEREOF IKZF3, ZC3HAV1L, CXXC5 CYP1A2 1723/4885ALDH1A1 3409/4885TSHR 2758/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.