SCHEMBL4137510

SCHEMBL4137510

COc1ccc2nccc(CCC3(O)CCC4(CC3)CN(c3ccc5c(c3)OCCO5)C(=O)O4)c2n1

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 12/20 0.43
SSTR5 P35346 1/20 0.35
SLC2A1 P11166 1/20 0.35
CLK1 P49759 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2254016 1.00 KCNH2 (0.43) KCNH2SSTR5SLC2A1CLK1
SCHEMBL2250556 1.00 KCNH2 (0.43) KCNH2SSTR5SLC2A1CLK1
SCHEMBL2250560 1.00 KCNH2 (0.43) KCNH2SSTR5SLC2A1CLK1
SCHEMBL2256847 0.88 KCNH2 (0.49) KCNH2
SCHEMBL2252556 0.88 KCNH2 (0.49) KCNH2
SCHEMBL2252560 0.88 KCNH2 (0.49) KCNH2
SCHEMBL2253508 0.83 KCNH2 (0.39) KCNH2
SCHEMBL2255530 0.83 KCNH2 (0.39) KCNH2
SCHEMBL2253511 0.83 KCNH2 (0.39) KCNH2
SCHEMBL3154178 0.82 KCNH2 (0.35) KCNH2SSTR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2066678-A1 SPIRO ANTIBIOTIC DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2009-06-10 EP claimed
WO-2008026172-A1 SPIRO ANTIBIOTIC DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-03-06 WO claimed
EP-2066678-A1 SPIRO ANTIBIOTIC DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2009-06-10 EP disclosed
WO-2008026172-A1 SPIRO ANTIBIOTIC DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-03-06 WO disclosed