SCHEMBL4150347

SCHEMBL4150347

CSc1ccc(NC(=O)c2c(C(C)C)csc2NC(=O)C(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ANO1 Q5XXA6 10/20 0.41
TP53 P04637 2/20 0.41
MAPT P10636 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ANO2 Q9NQ90 1/20 0.38
ABCC1 P33527 1/20 0.36
FPR2 P25090 1/20 0.36
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
PTGS2 P35354 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4146082 0.91 ANO1 (0.36) ANO1TP53MAPTSMN1; SMN2ANO2
SCHEMBL4147196 0.86 ANO1 (0.53) ANO1TP53MAPTSMN1; SMN2ANO2
SCHEMBL4149999 0.78 KMT2A (0.50) TP53MAPTSMN1; SMN2
SCHEMBL4147437 0.78 POLB (0.49) ANO1TP53MAPTSMN1; SMN2
SCHEMBL4141063 0.77 ABCC1 (0.56) ANO1MAPTSMN1; SMN2ABCC1
SCHEMBL1774979 0.75 MAPT (0.54) TP53MAPTSMN1; SMN2PTGS2
SCHEMBL4135342 0.73 BRD4 (0.49) ANO1TP53MAPTSMN1; SMN2
SCHEMBL4139676 0.72 ANO1 (0.78) ANO1TP53MAPTSMN1; SMN2ANO2
SCHEMBL4150055 0.72 ABCC1 (0.40) TP53MAPTABCC1
SCHEMBL4148960 0.71 TP53 (0.79) ANO1TP53MAPTSMN1; SMN2ANO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090143411-A1 Thiophens and Their Use as Anti-Tumor Agents COMPASS PHARMACEUTICALS LLC (US) 2009-06-04 US claimed
EP-1802634-A2 THIOPHENS AND THEIR USE AS ANTI-TUMOR AGENTS Compass Pharmaceuticals LLC (US) 2007-07-04 EP claimed
WO-2006044826-A2 THIOPHENS AND THEIR USE AS ANTI-TUMOR AGENTS COMPASS PHARMACEUTICALS LLC (US) 2006-04-27 WO claimed
US-20090143411-A1 Thiophens and Their Use as Anti-Tumor Agents COMPASS PHARMACEUTICALS LLC (US) 2009-06-04 US disclosed
EP-1802634-A2 THIOPHENS AND THEIR USE AS ANTI-TUMOR AGENTS Compass Pharmaceuticals LLC (US) 2007-07-04 EP disclosed
WO-2006044826-A2 THIOPHENS AND THEIR USE AS ANTI-TUMOR AGENTS COMPASS PHARMACEUTICALS LLC (US) 2006-04-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090143411-A1 Thiophens and Their Use as Anti-Tumor Agents TP53, BRDT, VHL ANO1 3854/4885TP53 1/4885MAPT 1629/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.