SCHEMBL4152290

SCHEMBL4152290

CN(C)CCNc1ccc(-c2nc3c(C(=O)NC(C)(C)C)ccnc3[nH]2)cc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 1/20 0.44
UHRF1 Q96T88 1/20 0.44
GSK3B P49841 5/20 0.39
SYK P43405 5/20 0.37
RIPK1 Q13546 1/20 0.36
PARP1 P09874 4/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
POLB P06746 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CDC7 O00311 1/20 0.35
CDK19 Q9BWU1 1/20 0.35
HDAC2 Q92769 1/20 0.35
ATAD2 Q6PL18 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4157285 0.92 RAD52 (0.42) RAD52UHRF1GSK3BSYKPARP1
SCHEMBL4147748 0.92 RAD52 (0.42) RAD52UHRF1GSK3BSYKPARP1
SCHEMBL4162859 0.91 RAD52 (0.42) RAD52UHRF1GSK3BSYKPARP1
SCHEMBL4961738 0.87 RAD52 (0.43) RAD52UHRF1GSK3BPARP1KDM4E
SCHEMBL4144903 0.85 RAD52 (0.46) RAD52UHRF1GSK3BKDM4ENPC1
SCHEMBL4157347 0.85 RAD52 (0.41) RAD52UHRF1GSK3BPARP1KDM4E
SCHEMBL4160387 0.85 RAD52 (0.43) RAD52UHRF1GSK3BPARP1KDM4E
SCHEMBL4161286 0.84 RAD52 (0.42) RAD52UHRF1GSK3BPARP1KDM4E
SCHEMBL4144891 0.83 RAD52 (0.42) RAD52UHRF1KDM4ERAB9A
SCHEMBL4152071 0.82 RAD52 (0.41) RAD52UHRF1GSK3BPARP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090170847-A1 Imidazopyridine Derivatives Inhibiting Protein Kinase Activity, Method for the Preparation Thereof and Pharmaceutical Composition Containing Same YUYU PHARMA, INC. (KR) 2009-07-02 US claimed
EP-1984370-A1 IMIDAZOPYRIDINE DERIVATIVES INHIBITING PROTEIN KINASE ACTIVITY, METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING SAME Crystalgenomics, Inc. (KR) 2008-10-29 EP claimed
WO-2007083978-A1 IMIDAZOPYRIDINE DERIVATIVES INHIBITING PROTEIN KINASE ACTIVITY, METHOD FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING SAME CRYSTALGENOMICS, INC. (KR) 2007-07-26 WO claimed
US-20090170847-A1 Imidazopyridine Derivatives Inhibiting Protein Kinase Activity, Method for the Preparation Thereof and Pharmaceutical Composition Containing Same YUYU PHARMA, INC. (KR) 2009-07-02 US disclosed
US-20090170847-A1 Imidazopyridine Derivatives Inhibiting Protein Kinase Activity, Method for the Preparation Thereof and Pharmaceutical Composition Containing Same YUYU PHARMA, INC. (KR) 2009-07-02 US disclosed
US-20090170847-A1 Imidazopyridine Derivatives Inhibiting Protein Kinase Activity, Method for the Preparation Thereof and Pharmaceutical Composition Containing Same YUYU PHARMA, INC. (KR) 2009-07-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090170847-A1 Imidazopyridine Derivatives Inhibiting Protein Kinase Activity, Method for the Preparation Thereof and Pharmaceutical Composition Containing Same GSK3B, GSK3A, MAP3K3 RAD52 4618/4885UHRF1 3834/4885GSK3B 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.