Pyrazole

Pyrazole

SCHEMBL4166278

COc1cc(N2CCN(C(=O)Cn3nc(-n4cccn4)c(Cl)c3C)CC2)ccc1Cl.c1cn[nH]c1

nearest known ligand 0.64

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 20/20 0.64
CYP2C19 P33261 1/20 0.60
KCNH2 Q12809 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3465885 0.94 CCR1 (0.71) CCR1CYP2C19KCNH2
Pyrazole SCHEMBL4564639 0.89 CCR1 (0.63) CCR1CYP2C19KCNH2
Pyrazole SCHEMBL4564640 0.89 CCR1 (0.63) CCR1CYP2C19KCNH2
SCHEMBL3465511 0.83 CCR1 (0.71) CCR1CYP2C19KCNH2
SCHEMBL3465142 0.83 CCR1 (0.74) CCR1CYP2C19KCNH2
SCHEMBL3466240 0.82 CCR1 (0.69) CCR1CYP2C19KCNH2
SCHEMBL3466237 0.82 CCR1 (0.69) CCR1CYP2C19KCNH2
SCHEMBL3465797 0.82 CCR1 (0.73) CCR1CYP2C19KCNH2
SCHEMBL3879906 0.82 CCR1 (0.58) CCR1CYP2C19KCNH2
SCHEMBL3464305 0.81 CCR1 (0.79) CCR1CYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1691810-A4 SUBSTITUTED PIPERAZINES CHEMOCENTRYX INC (US) 2009-07-01 EP disclosed
EP-1691810-A1 SUBSTITUTED PIPERAZINES ChemoCentryx Inc (US) 2006-08-23 EP disclosed
WO-2005056015-A1 SUBSTITUTED PIPERAZINES CHEMOCENTRYX, INC. (US) 2005-06-23 WO disclosed