SCHEMBL4167384

SCHEMBL4167384

Cc1ccc2[nH]c3c(c2c1)CC(=O)Nc1ccc(I)cc1-3

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 20/20 0.75
CDK5 Q00535 16/20 0.75
CDK5R1 Q15078 16/20 0.75
CCNB2 O95067 16/20 0.75
CDK1 P06493 16/20 0.75
CCNB1 P14635 16/20 0.75
CCNB3 Q8WWL7 16/20 0.75
GSK3A P49840 5/20 0.58
KDM4E B2RXH2 1/20 0.53
MEN1 O00255 1/20 0.53
CDC7 O00311 1/20 0.53
PLK4 O00444 1/20 0.53
CHEK1 O14757 1/20 0.53
AURKA O14965 1/20 0.53
NPC1 O15118 1/20 0.53
PDPK1 O15530 1/20 0.53
CCNT1 O60563 1/20 0.53
CCNT2 O60583 1/20 0.53
ROCK2 O75116 1/20 0.53
GMNN O75496 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14488716 0.91 GSK3B (0.81) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL5688936 0.86 GSK3B (1.00) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL17481541 0.86 GSK3B (0.84) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL30319854 0.86 GSK3B (1.00) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL4177498 0.85 GSK3B (0.80) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL5690374 0.85 GSK3B (1.00) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL30319783 0.85 GSK3B (1.00) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL30319796 0.84 GSK3B (1.00) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL5688227 0.84 GSK3B (1.00) GSK3BCDK5CDK5R1CCNB2CDK1
SCHEMBL17481536 0.84 GSK3B (0.78) GSK3BCDK5CDK5R1CCNB2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009010298-A2 PAULLONE DERIVATIVES AND ITS USE TECHNISCHE UNIVERSITÄT CAROLO-WILHELMINA ZU BRAUNSCHWEIG (DE) 2009-01-22 WO disclosed