SCHEMBL4167628

SCHEMBL4167628

COc1cc2ncnc(Oc3cnc(CC(=O)O)c(OC)c3)c2cc1OC

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LCK P06239 2/20 0.57
KDR P35968 11/20 0.54
CSF1R P07333 3/20 0.53
PDGFRA P16234 1/20 0.53
RET P07949 1/20 0.52
KIF5B P33176 1/20 0.52
BRAF P15056 3/20 0.52
RAF1 P04049 2/20 0.50
PDGFRB P09619 4/20 0.49
FLT4 P35916 4/20 0.49
FLT3 P36888 3/20 0.49
EGFR P00533 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4168769 0.95 KDR (0.52) LCKKDRCSF1RPDGFRARET
SCHEMBL4170739 0.95 KDR (0.52) LCKKDRCSF1RPDGFRARET
SCHEMBL4175668 0.90 LCK (0.56) LCKKDRCSF1RPDGFRARET
SCHEMBL4178009 0.83 KDR (0.58) LCKKDRCSF1RPDGFRARET
SCHEMBL4508946 0.82 PDGFRB (0.61) KDRCSF1RPDGFRAPDGFRBFLT3
SCHEMBL1097542 0.82 PDGFRB (0.64) LCKKDRCSF1RPDGFRARET
SCHEMBL1097832 0.81 PDGFRB (0.67) KDRCSF1RPDGFRAPDGFRBFLT4
SCHEMBL4179204 0.80 PDGFRB (0.57) KDRCSF1RPDGFRABRAFRAF1
SCHEMBL4179313 0.80 PDGFRB (0.57) KDRCSF1RPDGFRAPDGFRBFLT4
SCHEMBL4161085 0.80 PDGFRB (0.77) KDRCSF1RBRAFRAF1PDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090233950-A1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2009-09-17 US disclosed
EP-1994023-A1 QUINAZOLINE DERIVATIVES AstraZeneca AB (SE) 2008-11-26 EP disclosed
WO-2007099317-A1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2007-09-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090233950-A1 QUINAZOLINE DERIVATIVES NQO2, CCNI, F12 LCK 1627/4885KDR 2384/4885CSF1R 666/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.