SCHEMBL4168264

SCHEMBL4168264

CC(=O)c1cccc(-c2ccc([C@H]3OCC[C@H]3NS(=O)(=O)C(C)C)cc2)c1

nearest known ligand 0.68

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRIA2 P42262 14/20 0.68
KCNH2 Q12809 9/20 0.66
KDM1A O60341 2/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
GRIA4 P48058 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4168267 1.00 GRIA2 (0.68) GRIA2KCNH2KDM1AALDH1A1LMNA
SCHEMBL4168262 1.00 GRIA2 (0.68) GRIA2KCNH2KDM1AALDH1A1LMNA
SCHEMBL4097619 0.81 GRIA2 (1.00) GRIA2KCNH2KDM1A
SCHEMBL4097616 0.81 GRIA2 (1.00) GRIA2KCNH2KDM1A
SCHEMBL4097607 0.81 GRIA2 (1.00) GRIA2KCNH2KDM1A
SCHEMBL4168112 0.80 GRIA2 (0.48) GRIA2KCNH2GRIA4
SCHEMBL4168115 0.80 GRIA2 (0.48) GRIA2KCNH2GRIA4
SCHEMBL4168109 0.80 GRIA2 (0.48) GRIA2KCNH2GRIA4
SCHEMBL4958828 0.79 GRIA2 (1.00) GRIA2KCNH2
SCHEMBL2187890 0.78 GRIA4 (0.55) GRIA2KCNH2GRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090170902-A1 COMPOUNDS WHICH POTENTIATE GLUTAMATE RECEPTOR AND USES THEREOF IN MEDICINE GLAXO GROUP LIMITED (GB) 2009-07-02 US claimed
EP-4584250-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS Biohaven Therapeutics Ltd. (VG) 2025-07-16 EP disclosed
WO-2024054811-A1 COMBINATION THERAPIES INCLUDING METAL CHANNEL ACTIVATORS BIOHAVEN THERAPEUTICS LTD. (VG) 2024-03-14 WO disclosed
US-20090170902-A1 COMPOUNDS WHICH POTENTIATE GLUTAMATE RECEPTOR AND USES THEREOF IN MEDICINE GLAXO GROUP LIMITED (GB) 2009-07-02 US disclosed
US-20090170902-A1 COMPOUNDS WHICH POTENTIATE GLUTAMATE RECEPTOR AND USES THEREOF IN MEDICINE GLAXO GROUP LIMITED (GB) 2009-07-02 US disclosed
US-20090170902-A1 COMPOUNDS WHICH POTENTIATE GLUTAMATE RECEPTOR AND USES THEREOF IN MEDICINE GLAXO GROUP LIMITED (GB) 2009-07-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090170902-A1 COMPOUNDS WHICH POTENTIATE GLUTAMATE RECEPTOR AND USES THEREOF IN MEDICINE GRIN1, GRM1, GRIN2C GRIA2 16/4885KCNH2 1455/4885KDM1A 2792/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.