SCHEMBL4172018

SCHEMBL4172018

CC(C)(C)C(=O)CS(=O)(=O)C(C)(C)C(=O)Nc1cc(C(C)(C)C)on1.CC(C)(C)C(=O)CS(=O)(=O)C(C)(C)C(=O)Nc1ccc(C(F)(F)F)cn1

nearest known ligand 0.68

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 15/20 0.68
CNR1 P21554 11/20 0.68
CYP2C8 P10632 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
EGFR P00533 1/20 0.41
NPY5R Q15761 1/20 0.41
HPGD P15428 1/20 0.40
MAPK14 Q16539 1/20 0.40
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1620771 0.90 CNR1 (0.51) CNR2CNR1NPY5RGAA
SCHEMBL1621406 0.85 CNR2 (0.58) CNR2CNR1EGFRHPGDMAPK14
SCHEMBL1464269 0.81 CNR2 (1.00) CNR2CNR1CYP2C8CYP2D6CYP2C19
SCHEMBL4013229 0.81 CNR2 (0.56) CNR2CNR1CYP2C8CYP2D6CYP2C19
SCHEMBL2254622 0.79 CNR2 (0.66) CNR2CNR1CYP2C8CYP2D6CYP2C19
SCHEMBL4011949 0.79 CNR2 (0.55) CNR2CNR1CYP2C8CYP2D6CYP2C19
SCHEMBL3658651 0.78 CNR2 (0.58) CNR2CNR1CYP2C8CYP2D6CYP2C19
SCHEMBL3968895 0.77 CNR2 (0.67) CNR2CNR1NPY5R
SCHEMBL1463732 0.76 CNR2 (1.00) CNR2CNR1CYP2C8CYP2D6CYP2C19
SCHEMBL1621448 0.76 CNR1 (0.49) CNR2CNR1NPY5RGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074084-A1 COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR Boehringer Ingelheim International GmbH (DE) 2009-07-01 EP disclosed
WO-2008039645-A1 COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-04-03 WO disclosed