SCHEMBL4186295

SCHEMBL4186295

CCS(=O)(=O)N1CCN(CCCCCCCCCn2c(C)c(C)c3c4c(Cl)cc(=O)[nH]c4ccc32)CC1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.47
HTR7 P34969 6/20 0.38
HTR1A P08908 1/20 0.37
THRB P10828 8/20 0.36
CNR1 P21554 1/20 0.36
KMT2A Q03164 1/20 0.34
CHRM1 P11229 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4180698 0.79 AR (0.46) ARHTR1ATHRBCNR1KMT2A
SCHEMBL4182827 0.79 AR (0.49) AR
SCHEMBL4151770 0.78 AR (0.54) ARKMT2A
SCHEMBL4138453 0.77 AR (0.62) ARKMT2A
SCHEMBL4140291 0.76 AR (0.56) ARKMT2A
SCHEMBL4179098 0.76 AR (0.47) ARKMT2A
SCHEMBL4175644 0.75 AR (0.42) AR
SCHEMBL13697911 0.75 AR (0.38) ARKMT2A
SCHEMBL4183090 0.74 AR (0.41) AR
SCHEMBL4178893 0.74 AR (0.41) AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090227571-A1 Androgen Receptor Modulator Compounds and Methods LIGAND PHARMACEUTICALS INCORPORATED 2009-09-10 US claimed
US-20090227571-A1 Androgen Receptor Modulator Compounds and Methods LIGAND PHARMACEUTICALS INCORPORATED 2009-09-10 US disclosed
US-20090227571-A1 Androgen Receptor Modulator Compounds and Methods LIGAND PHARMACEUTICALS INCORPORATED 2009-09-10 US disclosed
US-20090227571-A1 Androgen Receptor Modulator Compounds and Methods LIGAND PHARMACEUTICALS INCORPORATED 2009-09-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090227571-A1 Androgen Receptor Modulator Compounds and Methods AR, NR5A1, ESRRA AR 1/4885HTR7 359/4885HTR1A 488/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.