SCHEMBL4187231

SCHEMBL4187231

Cc1nc(NC(=O)CCc2ccccc2)sc1C(=O)O

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.76
RXFP1 Q9HBX9 2/20 0.60
ADORA3 P0DMS8 1/20 0.58
MAOB P27338 1/20 0.58
ADORA2A P29274 1/20 0.58
ADORA2B P29275 1/20 0.58
ADORA1 P30542 1/20 0.58
PKM P14618 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
SCD O00767 1/20 0.58
RAB9A P51151 5/20 0.57
ALDH1A1 P00352 3/20 0.57
KMT2A Q03164 2/20 0.56
MEN1 O00255 1/20 0.54
POLB P06746 3/20 0.54
MAPT P10636 2/20 0.54
CSNK1D P48730 1/20 0.54
KDM4E B2RXH2 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12271557 0.88 NPC1 (0.61) NPC1RXFP1ADORA3MAOBADORA2A
SCHEMBL3579438 0.87 SCD (0.79) NPC1RXFP1ADORA3MAOBADORA2A
SCHEMBL27706943 0.86 NPC1 (0.62) NPC1RXFP1ADORA3MAOBADORA2A
SCHEMBL773084 0.83 LCK (0.71) NPC1SCDRAB9AALDH1A1SMN1; SMN2
SCHEMBL525062 0.81 NPC1 (1.00) NPC1PKMTDP1RAB9AALDH1A1
SCHEMBL15634098 0.81 CSNK1D (0.79) NPC1RXFP1PKMTDP1SCD
SCHEMBL28773945 0.81 NPC1 (0.56) NPC1RXFP1ADORA3MAOBADORA2A
SCHEMBL27706877 0.80 NPC1 (0.55) NPC1RXFP1ADORA3MAOBADORA2A
SCHEMBL3593815 0.80 SCD (0.76) NPC1RXFP1ADORA3MAOBADORA2A
SCHEMBL12443650 0.80 NPC1 (0.87) NPC1RXFP1RAB9AALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029138-A1 AMINOTHIAZOLE DERIVATIVES AS HUMAN STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2009-03-04 EP disclosed
WO-2007130075-A1 AMINOTHIAZOLE DERIVATIVES AS HUMAN STEAROYL-COA DESATURASE INHIBITORS XENON PHARMACEUTICALS INC. (CA) 2007-11-15 WO disclosed