SCHEMBL4187870

SCHEMBL4187870

O=C(O)Nc1ccc(-c2nc(C3=CCOCC3)c3cnn(CC(F)(F)F)c3n2)cc1

nearest known ligand 0.83

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 20/20 0.83
MTOR P42345 20/20 0.83
PIK3CD O00329 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4170362 0.93 PIK3CA (0.87) PIK3CAMTORPIK3CD
SCHEMBL4181215 0.92 PIK3CA (0.82) PIK3CAMTORPIK3CD
SCHEMBL7876645 0.92 PIK3CA (0.85) PIK3CAMTORPIK3CD
SCHEMBL4170322 0.91 PIK3CA (1.00) PIK3CAMTORPIK3CD
SCHEMBL4183872 0.90 PIK3CA (0.85) PIK3CAMTORPIK3CD
SCHEMBL4173217 0.89 MTOR (0.79) PIK3CAMTORPIK3CD
SCHEMBL4180309 0.89 PIK3CA (1.00) PIK3CAMTORPIK3CD
SCHEMBL4187812 0.88 PIK3CA (0.75) PIK3CAMTORPIK3CD
SCHEMBL4185067 0.88 PIK3CA (1.00) PIK3CAMTOR
Trifluoroacetic Acid SCHEMBL4182876 0.86 PIK3CA (0.94) PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009097490-A1 1H-PYRAZOLO[3,4-D]PYRIMIDINE, PURINE, 7H-PURIN-8(9H)-ONE, 3H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDINE, AND THIENO[3,2-D]PYRIMIDINE COMPOUNDS, THEIR USE AS mTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH (US) 2009-08-06 WO claimed
WO-2009097490-A1 1H-PYRAZOLO[3,4-D]PYRIMIDINE, PURINE, 7H-PURIN-8(9H)-ONE, 3H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDINE, AND THIENO[3,2-D]PYRIMIDINE COMPOUNDS, THEIR USE AS mTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH (US) 2009-08-06 WO disclosed