SCHEMBL4188601

SCHEMBL4188601

CCOc1cc(-c2nc(SCC(=O)NC(C)C)nc3[nH]cc(C#N)c23)c(Cl)cc1OC

nearest known ligand 0.81

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 13/20 0.81
HSP90AA1 P07900 3/20 0.72
KCNH2 Q12809 5/20 0.60
SMN1; SMN2 Q16637 2/20 0.42
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3956737 0.95 HSP90AB1 (0.89) HSP90AB1HSP90AA1KCNH2SMN1; SMN2
SCHEMBL3953828 0.91 HSP90AB1 (0.85) HSP90AB1HSP90AA1KCNH2SMN1; SMN2
SCHEMBL3961384 0.91 HSP90AB1 (0.92) HSP90AB1HSP90AA1KCNH2
SCHEMBL3962315 0.90 HSP90AB1 (1.00) HSP90AB1HSP90AA1KCNH2SMN1; SMN2
SCHEMBL13905698 0.89 HSP90AB1 (0.81) HSP90AB1HSP90AA1KCNH2SMN1; SMN2
SCHEMBL3962983 0.88 HSP90AB1 (0.74) HSP90AB1HSP90AA1KCNH2
SCHEMBL3958250 0.86 HSP90AB1 (1.00) HSP90AB1HSP90AA1KCNH2
SCHEMBL3955711 0.84 HSP90AB1 (0.80) HSP90AB1HSP90AA1KCNH2
SCHEMBL3950788 0.84 HSP90AA1 (1.00) HSP90AB1HSP90AA1KCNH2SMN1; SMN2
SCHEMBL3958501 0.84 HSP90AB1 (0.74) HSP90AB1HSP90AA1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009030871-A1 PYRROLOPYRIMIDINE DERIVATIVES HAVING HSP90 INHIBITORY ACTIVITY VERNALIS R & D LTD (GB) 2009-03-12 WO claimed
WO-2009030871-A1 PYRROLOPYRIMIDINE DERIVATIVES HAVING HSP90 INHIBITORY ACTIVITY VERNALIS R & D LTD (GB) 2009-03-12 WO disclosed
WO-2009030871-A1 PYRROLOPYRIMIDINE DERIVATIVES HAVING HSP90 INHIBITORY ACTIVITY VERNALIS R & D LTD (GB) 2009-03-12 WO disclosed