SCHEMBL4189173

SCHEMBL4189173

COc1cccc(CCc2ccccc2O)c1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 15/20 0.62
HTR1A P08908 3/20 0.62
DRD2 P14416 3/20 0.62
ABCG2 Q9UNQ0 1/20 0.61
TAAR1 Q96RJ0 1/20 0.56
GABRA1 P14867 1/20 0.54
GABRG2 P18507 1/20 0.54
GABRB3 P28472 1/20 0.54
GABRA3 P34903 1/20 0.54
GABRA2 P47869 1/20 0.54
GABRB2 P47870 1/20 0.54
CYP2D6 P10635 1/20 0.53
HTR2A P28223 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30416326 1.00 ABCB1 (0.62) ABCB1HTR1ADRD2ABCG2TAAR1
SCHEMBL19900978 0.91 ESR1 (0.56) ABCB1HTR1ADRD2ABCG2TAAR1
SCHEMBL8702673 0.91 CHRM2 (0.54) ABCB1HTR1ADRD2ABCG2TAAR1
SCHEMBL19900980 0.89 HDAC1 (0.56) ABCB1HTR1ADRD2ABCG2TAAR1
SCHEMBL19900867 0.89 HDAC1 (0.56) ABCB1HTR1ADRD2ABCG2TAAR1
SCHEMBL19900804 0.89 HDAC1 (0.56) ABCB1HTR1ADRD2ABCG2TAAR1
SCHEMBL19900723 0.89 HDAC1 (0.56) ABCB1HTR1ADRD2ABCG2TAAR1
SCHEMBL19900758 0.89 HDAC1 (0.56) ABCB1HTR1ADRD2ABCG2TAAR1
SCHEMBL19900816 0.89 HDAC1 (0.56) ABCB1HTR1ADRD2ABCG2TAAR1
SCHEMBL8704118 0.87 AKR1B1 (0.60) ABCB1HTR1ADRD2ABCG2GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 54 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200375949-A1 BISPHENOL COMPOUNDS TEMPLE UNIVERSITY - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2020-12-03 US claimed
CN-111807976-A Novel method for preparing sarpogrelate hydrochloride 深圳市道科思医药有限公司 2020-10-23 CN claimed
WO-2019104153-A1 BISPHENOL COMPOUNDS THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2019-05-31 WO claimed
CN-105906486-B The synthetic method of Sarpogrelate intermediate 2 [2 (3 methoxyphenyl) ethyl] phenol 安徽修制药有限公司 2018-04-20 CN claimed
CN-105906486-A Synthetic method of sarpogrelate intermediate 2-[2-(3-methoxyphenyl)ethyl]phenol 安徽禾益化学股份有限公司 2016-08-31 CN claimed
CN-103965063-B Sarpogrelate hydrochloride new preparation process Limited liability company of Kechuang institute of materia medica, Anhui (CN) 2016-05-25 CN claimed
EP-3503879-B1 COMPOSITION COMPRISING (A) A DUAL AGENT ACTING AS A 5-HT2A RECEPTOR ANTAGONIST AND CYP2D6 INHIBITOR AND (B) AN NMDA RECEPTOR ANTAGONIST FOR USE IN THE TREATMENT OF DISEASES INVOLVING GLUCOSE Exciva GmbH (DE) 2026-04-22 EP disclosed
US-20250216782-A1 MASKING PROCESS USING SWITCHABLE POLYMER TOKYO ELECTRON LTD (JP) 2025-07-03 US disclosed
CN-117964462-A Preparation method of 1-benzyloxy-2- [2- (3-methoxyphenyl) vinyl ] benzene 苏州诚和医药化学有限公司 2024-05-03 CN disclosed
CN-110831584-B Targeted drug rescue with novel compositions, combinations and methods thereof 埃克塞瓦有限责任公司 2023-03-10 CN disclosed
US-11478467-B2 Targeted drug rescue with novel compositions, combinations, and methods thereof Exciva GmbH (DE) 2022-10-25 US disclosed
US-20210228508-A1 COMPOSITIONS AND METHODS THEREOF Exciva GmbH 2021-07-29 US disclosed
US-20210228508-A1 COMPOSITIONS AND METHODS THEREOF Exciva GmbH 2021-07-29 US disclosed
CN-1245426-A Composition containing diarylalkane derivative as effective component for treating or preventing pancreatitis SANKYO CO (JP) 2000-02-23 CN disclosed
EP-0958817-A1 COMPOSITION CONTAINING DIARYLALKANE DERIVATIVE AS THE ACTIVE INGREDIENT FOR TREATING OR PREVENTING PANCREATITIS SANKYO COMPANY LIMITED (JP) 1999-11-24 EP disclosed
CN-1044365-C Alpha, omega-diarylalkane derivatives, their preparation and their use in the treatment and prevention of circulatory diseases and psychosis SANKYO CO (JP) 1999-07-28 CN disclosed
EP-0844000-A1 Use of alpha, omega-diarylalkane derivatives in the treatment and prevention of psychosis SANKYO COMPANY LIMITED (JP) 1998-05-27 EP disclosed
US-5556864-A TREATMENT OF CIRCULATORY DISEASES AND PSYCHOSIS SANKYO COMPANY, LIMITED (JP) 1996-09-17 US disclosed
CN-1102640-A Alpha, omega-diarylalkane derivatives, their preparation and their use in the treatment and prevention of circulatory and psychiatric disorders SANKYO CO (JP) 1995-05-17 CN disclosed
EP-0600717-A1 Phenoxyalkylamines, -pyrrolidines and -piperidines for the treatment and prevention of circulatory diseases and psychosis SANKYO COMPANY LIMITED (JP) 1994-06-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11478467-B2 Targeted drug rescue with novel compositions, combinations, and methods thereof HTR2A, HTR2C, CYP3A43 ABCB1 50/4885HTR1A 24/4885DRD2 262/4885
US-20200375949-A1 BISPHENOL COMPOUNDS RPP30, RPS10, RPS20 ABCB1 2054/4885HTR1A 3326/4885DRD2 2596/4885
US-20210228508-A1 COMPOSITIONS AND METHODS THEREOF CYP21A2, CYP2C19, CYP2F1 ABCB1 98/4885HTR1A 1544/4885DRD2 614/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.