SCHEMBL4209348

SCHEMBL4209348

CN1CCn2c(nc(-c3ccncc3)cc2=O)C(C(N)=O)C1

nearest known ligand 0.50

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 18/20 0.50
CYP1A2 P05177 3/20 0.41
CYP2D6 P10635 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4217864 0.88 GSK3B (0.41) GSK3BCYP1A2CYP2D6
SCHEMBL3658703 0.86 GSK3B (0.53) GSK3BCYP2D6
SCHEMBL4210550 0.84 GSK3B (0.54) GSK3BCYP1A2CYP2D6
SCHEMBL4380859 0.82 GSK3B (0.40) GSK3BCYP1A2CYP2D6
SCHEMBL4221005 0.81 ROCK1 (0.45) GSK3BCYP1A2CYP2D6
SCHEMBL3398094 0.80 GSK3B (0.39) GSK3BCYP1A2CYP2D6
SCHEMBL3658356 0.80 GSK3B (0.48) GSK3B
Hydrochloric Acid SCHEMBL4212507 0.79 GSK3B (0.47) GSK3BCYP2D6
SCHEMBL4391271 0.73 GSK3B (0.39) GSK3BCYP1A2CYP2D6
SCHEMBL4217866 0.73 GSK3B (0.42) GSK3BCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2238140-B1 SUBSTITUTED HETEROARYLAMIDE DIAZEPINOPYRIMIDONE DERIVATIVES SANOFI SA (FR) 2013-07-17 EP claimed
EP-2130922-A1 IMPROVED HALOHYDRIN EPOXIDASE Mitsubishi Rayon Co. Ltd. (JP) 2009-12-09 EP disclosed