SCHEMBL4212469

SCHEMBL4212469

Cc1ccnc(CNCCCC(N)Cc2ncc(C)cc2C)c1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 1/20 0.34
SCN8A Q9UQD0 1/20 0.33
KDM1A O60341 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
F2 P00734 3/20 0.32
CHRM2 P08172 1/20 0.32
SIRT2 Q8IXJ6 1/20 0.31
NOS1 P29475 2/20 0.30
SLC40A1 Q9NP59 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5574543 0.79 CXCR4 (0.36) CXCR4SCN8A
SCHEMBL4212477 0.76 CXCR4 (0.40) CXCR4KDM1AMAOAMAOB
SCHEMBL5576619 0.74 CXCR4 (0.32) CXCR4SLC40A1
SCHEMBL4206736 0.74 CXCR4 (0.42) CXCR4CHRM2NOS1
SCHEMBL10483857 0.72 CHRM2 (0.42) CXCR4SCN8AKDM1AMAOAMAOB
SCHEMBL10483874 0.72 KDM1A (0.43) SCN8AKDM1AMAOAMAOBCHRM2
SCHEMBL5574432 0.72 CXCR4 (0.48) CXCR4SCN8A
SCHEMBL5576023 0.71 SCN8A (0.38) CXCR4SCN8ACHRM2SIRT2SLC40A1
SCHEMBL23428545 0.71 CHRM2 (0.45) CXCR4SCN8AKDM1AMAOAMAOB
SCHEMBL3265517 0.71 CHRM2 (0.44) SCN8AKDM1AMAOAMAOBCHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed