SCHEMBL4213636

SCHEMBL4213636

Cc1cncc(CNCC(O)C(Cc2ccccc2)NC(=O)c2cccc(C(=O)N(C)Cc3nc(C)cs3)c2)c1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.49
CTSD P07339 9/20 0.46
BACE2 Q9Y5Z0 6/20 0.44
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4218559 1.00 BACE1 (0.49) BACE1CTSDBACE2CYP3A4
SCHEMBL4218447 0.94 BACE1 (0.51) BACE1CTSDBACE2CYP3A4
SCHEMBL4204587 0.94 BACE1 (0.51) BACE1CTSDBACE2CYP3A4
SCHEMBL4219051 0.93 BACE1 (0.48) BACE1CTSDBACE2CYP3A4
SCHEMBL3508855 0.93 BACE1 (0.48) BACE1CTSDBACE2CYP3A4
SCHEMBL3511559 0.93 BACE1 (0.48) BACE1CTSDBACE2
SCHEMBL3509365 0.93 BACE1 (0.48) BACE1CTSDBACE2CYP3A4
SCHEMBL4208740 0.93 BACE1 (0.48) BACE1CTSDBACE2CYP3A4
SCHEMBL3509801 0.93 BACE1 (0.48) BACE1CTSDBACE2CYP3A4
SCHEMBL3510513 0.93 BACE1 (0.48) BACE1CTSDBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504420-B2 Compounds which inhibit beta-secretase activity and methods of use COMENTIS, INC. (US) 2009-03-17 US claimed