SCHEMBL4215633

SCHEMBL4215633

CC(C)(C)OC(=O)N1CC(O)C2NCC[C@H]21

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.42
CHRM1 P11229 1/20 0.42
CHRM3 P20309 1/20 0.42
AR P10275 1/20 0.34
HSD17B10 Q99714 1/20 0.34
NR1H2 P55055 1/20 0.33
CYP1A2 P05177 1/20 0.33
POLB P06746 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
PREP P48147 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13944478 1.00 CHRM2 (0.42) CHRM2CHRM1CHRM3ARHSD17B10
SCHEMBL4050279 1.00 CHRM2 (0.42) CHRM2CHRM1CHRM3ARHSD17B10
SCHEMBL4191884 1.00 CHRM2 (0.42) CHRM2CHRM1CHRM3ARHSD17B10
SCHEMBL30723481 0.85 CHRM2 (0.41) CHRM2CHRM1CHRM3ARHSD17B10
SCHEMBL30723452 0.85 CHRM2 (0.41) CHRM2CHRM1CHRM3ARHSD17B10
SCHEMBL30723502 0.85 CHRM2 (0.41) CHRM2CHRM1CHRM3ARHSD17B10
SCHEMBL22949990 0.84 CHRM2 (0.38) CHRM2CHRM1CHRM3ARHSD17B10
SCHEMBL8350117 0.83 CHRM2 (0.40) CHRM2CHRM1CHRM3ARHSD17B10
SCHEMBL23273865 0.80 CHRM2 (0.41) CHRM2CHRM1CHRM3ARHSD17B10
SCHEMBL22587052 0.80 CHRM2 (0.41) CHRM2CHRM1CHRM3ARHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP disclosed
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed