SCHEMBL4225976

SCHEMBL4225976

CC(C)Oc1cc(CN2CCC(Nc3ncc(-c4ccccc4)cn3)CC2)cc(OC(C)C)c1.c1ccc(-c2cnc(NC3CCNCC3)nc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SSTR5 P35346 1/20 0.54
ACHE P22303 8/20 0.41
BACE1 P56817 5/20 0.41
HDAC1 Q13547 1/20 0.40
MAPK8 P45983 1/20 0.40
SIGMAR1 Q99720 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ROCK2 O75116 2/20 0.38
CCR2 P41597 1/20 0.38
ROCK1 Q13464 1/20 0.38
NSD2 O96028 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3787453 0.94 SSTR5 (0.59) SSTR5ACHEBACE1SIGMAR1KMT2A
SCHEMBL4236818 0.89 SSTR5 (0.47) SSTR5ACHEBACE1HDAC1SIGMAR1
SCHEMBL3781183 0.88 SSTR5 (0.52) SSTR5ACHEBACE1SIGMAR1
SCHEMBL4240279 0.87 SSTR5 (0.50) SSTR5ACHEBACE1MAPK8MEN1
SCHEMBL3774524 0.85 SSTR5 (0.53) SSTR5ACHEBACE1SIGMAR1ROCK2
SCHEMBL3785452 0.85 SSTR5 (0.52) SSTR5ACHEBACE1SIGMAR1MEN1
SCHEMBL4233983 0.85 SSTR5 (0.47) SSTR5ACHE
SCHEMBL3774157 0.83 SSTR5 (0.51) SSTR5ACHEBACE1SIGMAR1
SCHEMBL27756066 0.83 SSTR5 (0.49) SSTR5ACHEBACE1ROCK2CCR2
SCHEMBL3782674 0.81 SSTR5 (0.60) SSTR5ACHEBACE1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001867-B1 PYRIMIDINE, QUINAZOLINE, PTERIDINE AND TRIAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2009-07-01 EP disclosed
CN-101405284-A Pyrimidine, quinazoline, pteridine and derivatives HOFFMANN LA ROCHE (CH) 2009-04-08 CN disclosed