Acetic Acid

Acetic Acid

SCHEMBL4227622

CC(=O)O.O=C(/C=C/c1cnc(N[C@@H]2CCN(C(=O)O)C2)c(Cl)c1)NO

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Acetic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 2/20 0.40
HDAC1 Q13547 3/20 0.38
EHMT1 Q9H9B1 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
KDM5A P29375 1/20 0.38
EGFR P00533 1/20 0.37
CCNK O75909 9/20 0.37
CDK12 Q9NYV4 9/20 0.37
KCNH2 Q12809 1/20 0.36
MAPK3 P27361 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL4227631 1.00 JAK3 (0.40) JAK3HDAC1EHMT1HDAC6KDM5A
SCHEMBL4227861 0.97 JAK3 (0.38) JAK3HDAC1EHMT1HDAC6KDM5A
SCHEMBL4227848 0.97 JAK3 (0.38) JAK3HDAC1EHMT1HDAC6KDM5A
SCHEMBL4227627 0.88 JAK3 (0.37) JAK3KDM5AEGFRCCNKCDK12
Hydrochloric Acid SCHEMBL4227720 0.87 HDAC1 (0.45) JAK3HDAC1
Hydrochloric Acid SCHEMBL4227723 0.87 HDAC1 (0.45) JAK3HDAC1
Hydrochloric Acid SCHEMBL4861689 0.86 HDAC1 (0.47) HDAC1HDAC6MAPK3
Hydrochloric Acid SCHEMBL4227728 0.86 MAPK3 (0.47) JAK3HDAC1KCNH2MAPK3
Hydrochloric Acid SCHEMBL4227734 0.86 MAPK3 (0.47) JAK3HDAC1KCNH2MAPK3
Hydrochloric Acid SCHEMBL4223537 0.86 HDAC1 (0.45) HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7557127-B2 HDAC inhibitor ASTELLAS PHARMA INC. (JP) 2009-07-07 US disclosed
US-20090054464-A1 HDAC INHIBITOR ASTELLAS PHARMA INC. (JP) 2009-02-26 US disclosed
US-7465731-B2 HDAC inhibitor ASTELLAS PHARMA INC. (JP) 2008-12-16 US disclosed
US-20060052599-A1 HDAC inhibitor ASTELLAS PHARMA INC. (JP) 2006-03-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060052599-A1 HDAC inhibitor HDAC1, HDAC2, HDAC11 JAK3 4112/4885HDAC1 1/4885EHMT1 99/4885
US-20090054464-A1 HDAC INHIBITOR HDAC1, HDAC2, HDAC8 JAK3 4148/4885HDAC1 1/4885EHMT1 119/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.