SCHEMBL4245252

SCHEMBL4245252

CC(=O)NC(Cc1ccccc1)CC(O)CN(Cc1ccccc1)C(=O)OCc1cncs1

nearest known ligand 0.52

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 20/20 0.52
CYP2D6 P10635 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL894139 0.89 CYP3A4 (0.53) CYP3A4
SCHEMBL893483 0.85 TDP1 (0.50) CYP3A4CYP2D6
SCHEMBL4248588 0.84 CYP3A4 (0.49) CYP3A4CYP2D6
SCHEMBL4251990 0.84 CYP3A4 (0.61) CYP3A4CYP2D6
SCHEMBL4251351 0.82 CYP3A4 (0.44) CYP3A4CYP2D6
SCHEMBL893562 0.81 CYP3A4 (0.51) CYP3A4CYP2D6
SCHEMBL4251180 0.81 CYP3A4 (0.49) CYP3A4CYP2D6
SCHEMBL4959397 0.80 CYP3A4 (0.56) CYP3A4
SCHEMBL4959571 0.80 CYP3A4 (0.56) CYP3A4
SCHEMBL4390521 0.80 CYP3A4 (0.56) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP disclosed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO disclosed