SCHEMBL4246755

SCHEMBL4246755

C[C@@H]1CN(Cc2c[nH]nc2-c2cc[c]cc2)CCN1c1ccc(C(F)(F)F)cn1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SGPL1 O95470 3/20 0.41
CXCR3 P49682 6/20 0.38
SMO Q99835 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
LMNA P02545 1/20 0.36
KMT2A Q03164 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
HPGD P15428 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34
DRD4 P21917 1/20 0.34
GRM2 Q14416 1/20 0.34
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4398201 0.90 PTGDR2 (0.42) SGPL1CXCR3SMOSMN1; SMN2LMNA
SCHEMBL4244454 0.89 SGPL1 (0.41) SGPL1CXCR3SMOSMN1; SMN2LMNA
SCHEMBL14311334 0.89 SGPL1 (0.41) SGPL1CXCR3SMOSMN1; SMN2LMNA
SCHEMBL13592416 0.89 SGPL1 (0.41) SGPL1CXCR3SMOSMN1; SMN2LMNA
SCHEMBL13590836 0.89 SGPL1 (0.41) SGPL1CXCR3SMOSMN1; SMN2LMNA
SCHEMBL13590946 0.89 MAOB (0.45) SGPL1CXCR3SMO
SCHEMBL13590947 0.89 MAOB (0.45) SGPL1CXCR3SMO
SCHEMBL4249119 0.89 MAOB (0.45) SGPL1CXCR3SMO
SCHEMBL13590953 0.88 SGPL1 (0.40) SGPL1CXCR3SMOSMN1; SMN2LMNA
SCHEMBL4245413 0.88 SGPL1 (0.40) SGPL1CXCR3SMOSMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2057124-A2 COMPOUNDS AND COMPOSITIONS AS ITPKB INHIBITORS IRM, LLC (BM) 2009-05-13 EP disclosed
WO-2008011611-A2 COMPOUNDS AND COMPOSITIONS AS ITPKB INHIBITORS IRM LLC (BM) 2008-01-24 WO disclosed