SCHEMBL4248241

SCHEMBL4248241

O=C(O)COc1ccc2c(c1)S(=O)(=O)C=C(c1c(O)c3cc(F)ccc3n(Cc3ccc(F)cc3)c1=O)N2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.48
PIK3R1 P27986 1/20 0.38
PIK3CA P42336 1/20 0.38
NR1I2 O75469 1/20 0.38
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
BLM P54132 1/20 0.37
PMP22 Q01453 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PLA2G2A P14555 1/20 0.36
PTGDR2 Q9Y5Y4 6/20 0.36
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35
AKR1B1 P15121 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3920117 0.93 CYP2C9 (0.56) CYP2C9PIK3R1PIK3CANR1I2KDM4E
SCHEMBL3920627 0.92 CYP2C9 (0.47) CYP2C9PIK3R1PIK3CANR1I2KDM4E
SCHEMBL3919559 0.91 CYP2C9 (0.46) CYP2C9PIK3R1PIK3CANR1I2KDM4E
SCHEMBL3918627 0.91 CYP2C9 (0.46) CYP2C9PIK3R1PIK3CANR1I2KDM4E
SCHEMBL3930787 0.90 CYP2C9 (0.43) CYP2C9NR1I2KDM4EHDAC1HDAC8
SCHEMBL3922130 0.89 PIK3R1 (0.44) CYP2C9PIK3R1PIK3CANR1I2KDM4E
SCHEMBL3917989 0.86 CYP2C9 (0.42) CYP2C9PIK3R1PIK3CANR1I2KDM4E
SCHEMBL3929284 0.84 CYP2C9 (0.41) CYP2C9PIK3R1PIK3CANR1I2KDM4E
SCHEMBL3922914 0.84 CYP2C9 (0.39) CYP2C9PIK3R1PIK3CANR1I2KDM4E
SCHEMBL3920019 0.83 CYP2C9 (0.50) CYP2C9NR1I2KDM4ELMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1786807-B1 HETEROCYCLIC ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2009-07-29 EP claimed