SCHEMBL4251107

SCHEMBL4251107

NCCC(N)Cc1cnc2ccccc2c1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 2/20 0.47
CYP1A2 P05177 2/20 0.41
PDGFRB P09619 2/20 0.41
PDGFRA P16234 2/20 0.41
PDE10A Q9Y233 3/20 0.39
MMP1 P03956 1/20 0.39
FCER2 P06734 1/20 0.39
MMP3 P08254 1/20 0.39
MMP9 P14780 1/20 0.39
TPH1 P17752 1/20 0.39
KDM1A O60341 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
DHODH Q02127 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
DPP4 P27487 1/20 0.38
DPP8 Q6V1X1 1/20 0.38
MGAM O43451 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3936746 0.83 AKT1 (0.48) AKT1CYP1A2PDGFRBPDGFRAPDE10A
SCHEMBL22401385 0.80 HTR2A (0.57) AKT1CYP1A2PDGFRBPDGFRAPDE10A
SCHEMBL23009533 0.80 HTR2A (0.57) AKT1CYP1A2PDGFRBPDGFRAPDE10A
SCHEMBL3638034 0.77 DHODH (0.49) CYP1A2PDGFRBPDGFRAPDE10AKDM1A
SCHEMBL28270504 0.77 CYP1A2 (0.46) AKT1CYP1A2PDGFRBPDGFRAPDE10A
SCHEMBL263918 0.77 CYP1A2 (0.52) CYP1A2PDGFRBPDGFRAPDE10AKDM1A
SCHEMBL30101236 0.77 CYP1A2 (0.52) CYP1A2PDGFRBPDGFRAPDE10AKDM1A
SCHEMBL2267933 0.76 AKT1 (0.45) AKT1CYP1A2PDGFRBPDGFRAPDE10A
SCHEMBL2267925 0.76 CYP1A2 (0.44) AKT1CYP1A2PDGFRBPDGFRAPDE10A
SCHEMBL2267928 0.76 CYP1A2 (0.44) AKT1CYP1A2PDGFRBPDGFRAPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2081917-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF Abbott Laboratories (US) 2009-07-29 EP disclosed
WO-2008027932-A2 CYTOCHROME P450 OXIDASE INHIBITORS AND USES THEREOF ABBOTT LABORATORIES (US) 2008-03-06 WO disclosed